ホスホリラーゼ

  • 阻害剤の選択性比較
  • 溶解度
カタログ番号 製品カタログ 溶解度(25°C)
DMSO アルコール
S2717 CP-91149 <1 mg/mL 80 mg/mL <1 mg/mL
S2045 Doxifluridine 49 mg/mL 49 mg/mL <1 mg/mL
S3731 Tipiracil hydrochloride 55 mg/mL 8 mg/mL <1 mg/mL
製品コード 製品説明 文献中の使用例 お客様のフィードバック
S2717

CP-91149

CP-91149 is a selective glycogen phosphorylase (GP) inhibitor with IC50 of 0.13 μM in the presence of glucose, 5- to 10-fold less potent in the absence of glucose.

S2045

Doxifluridine

Doxifluridine is an oral prodrug that is converted to the cytotoxic agent 5-fluorouracil (5-FU).

S3731

Tipiracil hydrochloride

Tipiracil is an inhibitor of thymidine phosphorylase, the enzyme that degrades trifluridine into trifluorothymidine. Its combination with trifluridine increases the bioavailability of trifluridine.