Cyclothiazide

製品コードS6611 バッチS661101

化学情報

	Synonyms	N/A	Storage (From the date of receipt)	3 years -20°C powder
	化学式	C₁₄H₁₆ClN₃O₄S₂
	分子量	389.88	CAS No.	2259-96-3
Solubility (25°C)*	体外	DMSO	78 mg/mL (200.06 mM)
		Ethanol	19 mg/mL (48.73 mM)
		Water	Insoluble
* <1 mg/ml means slightly soluble or insoluble. * Please note that Selleck tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

溶剤液（一定の濃度）を調合する

生物活性

製品説明	Cyclothiazide is a positive allosteric modulator of ionotropic α-amino-3-hydroxy-5-methylisoxazole-4-propionic acid (AMPA)-type glutamate receptors with critical roles in neurological development and function.
in vitro	Cyclothiazide is known to produce a fast inhibition of AMPA receptor desensitization and a much slower potentiation of the AMPA current^[1].

プロトコル(参考用のみ)

参考

[1] Sergio Fucile, et al. Proc Natl Acad Sci U S A. 2006, 103(8): 2943–2947.

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長期の保管のために-20°Cの下で製品を保ってください。

人間や獣医の診断であるか治療的な使用のためにでない。

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