CPT

亜型選択性的な製品

CPT製品

  • All (5)
  • CPT阻害剤 (2)
  • CPT活性剤(1)
  • CPT作動薬(1)
  • 新製品
製品コード 製品名称 製品説明 文献中Selleckの製品使用例 お客様のフィードバック
S8244 Etomoxir sodium salt Etomoxir is an irreversible inhibitor of carnitine palmitoyltransferase-1 (CPT-1) on the outer face of the inner mitochondrial membrane. Etomoxir enhances palmitate-induced cell apoptosis.
Bioact Mater, 2024, 35:549-563
Oncogene, 2024, 43(6):406-419
Biochem Pharmacol, 2024, S0006-2952(24)00144-8
S9819 C75 C75 (4-Methylene-2-octyl-5-oxotetrahydrofuran-3-carboxylic acid) , a more stable synthetic mimic of cerulenin, inhibits fatty-acid synthase (FAS/FASN) with an IC50 of 15.53 μM and has potential therapeutic effects in several cancer models. C75 is also a potent CPT1A activator.
Theranostics, 2023, 13(13):4482-4496
Theranostics, 2023, 10.7150/thno.84921
Front Microbiol, 2022, 13:961942
S6959 Perhexiline maleate Perhexiline maleate is a potent inhibitor of carnitine palmitoyltransferase 1 (CPT1) with IC50s of 77 μM and 148 μM for rat heart CPT1 and liver CPT1, respectively, and also inhibits carnitine palmitoyltransferase 2 (CPT2).
Cancer Cell, 2022, S1535-6108(22)00312-9
S2269 Baicalin Baicalin is an inhibitor of prolyl oligopeptidase and also is an allosteric activator of carnitine palmityl transferase 1 (CPT1). Baicalin reduces the expression of NF-κB.
Chem Biol Interact, 2024, 387:110820
Int J Mol Sci, 2023, 24(11)9435
Molecules, 2021, 26(5)1210
S9819 C75 C75 (4-Methylene-2-octyl-5-oxotetrahydrofuran-3-carboxylic acid) , a more stable synthetic mimic of cerulenin, inhibits fatty-acid synthase (FAS/FASN) with an IC50 of 15.53 μM and has potential therapeutic effects in several cancer models. C75 is also a potent CPT1A activator.
Theranostics, 2023, 13(13):4482-4496
Theranostics, 2023, 10.7150/thno.84921
Front Microbiol, 2022, 13:961942
S8244 Etomoxir sodium salt Etomoxir is an irreversible inhibitor of carnitine palmitoyltransferase-1 (CPT-1) on the outer face of the inner mitochondrial membrane. Etomoxir enhances palmitate-induced cell apoptosis.
Bioact Mater, 2024, 35:549-563
Oncogene, 2024, 43(6):406-419
Biochem Pharmacol, 2024, S0006-2952(24)00144-8
S6959 Perhexiline maleate Perhexiline maleate is a potent inhibitor of carnitine palmitoyltransferase 1 (CPT1) with IC50s of 77 μM and 148 μM for rat heart CPT1 and liver CPT1, respectively, and also inhibits carnitine palmitoyltransferase 2 (CPT2).
Cancer Cell, 2022, S1535-6108(22)00312-9
S2269 Baicalin Baicalin is an inhibitor of prolyl oligopeptidase and also is an allosteric activator of carnitine palmityl transferase 1 (CPT1). Baicalin reduces the expression of NF-κB.
Chem Biol Interact, 2024, 387:110820
Int J Mol Sci, 2023, 24(11)9435
Molecules, 2021, 26(5)1210
S9819 C75 C75 (4-Methylene-2-octyl-5-oxotetrahydrofuran-3-carboxylic acid) , a more stable synthetic mimic of cerulenin, inhibits fatty-acid synthase (FAS/FASN) with an IC50 of 15.53 μM and has potential therapeutic effects in several cancer models. C75 is also a potent CPT1A activator.
Theranostics, 2023, 13(13):4482-4496
Theranostics, 2023, 10.7150/thno.84921
Front Microbiol, 2022, 13:961942

CPT阻害剤の選択性比較

Tags: CPT inhibitor|CPT agonist|CPT activator|CPT inducer|CPT antagonist|CPT signaling pathway|CPT assay kit