Degarelix acetate

製品コード：P1094 純度：99.94%

Degarelix acetate (ASP-3550 acetate) is a potent and long-acting luteinizing hormone-releasing hormone (LHRH) antagonist.

Amino-acid Sequence

CAS No. 214766-78-6

サイズ	価格(税別)	在庫状況
1mg	JPY 22300	国内在庫あり
5mg	JPY 67000	国内在庫あり
25mg	JPY 200800	お問い合わせ
100mg	JPY 502300	お問い合わせ
バルクサイズ	バルク特価あり

代表番号: 045-509-1970\|電子メール：[email protected] よく尋ねられる質問

現在のバッチを見る： P109401 DMSO] 33 mg/mL] false] Water] 33 mg/mL] false] Ethanol] Insoluble] false 純度： 99.94%

99.94

保管	3 years-20°C powder	溶液の保管冷凍と解凍の繰り返しを避けるため小分けにしてください	1年-80°Cin solvent
			1个月-20°Cin solvent

In vitro
Batch:

DMSO : 33 mg/mL ( (20.21 mM)；吸湿したDMSOは溶解度を減少させます。新しいDMSOをご使用ください。)

Water : 33 mg/mL

Ethanol : Insoluble

in vivo
Batch:

Add solvents to the product individually and in order.

製品説明	Degarelix acetate (ASP-3550 acetate) is a potent and long-acting luteinizing hormone-releasing hormone (LHRH) antagonist.

In Vivo
In vivo	Degarelix acetate is a member of a new class of long-acting gonadotropin-releasing hormone (GnRH) antagonists, possessing a long duration of luteinizing hormone (LH) and testosterone suppression.^[2]
動物実験	動物モデル	castrated male rat model
	投与量	50 μg
	投与経路	--

参考
[1] Broqua P, et al. J Pharmacol Exp Ther. 2002 Apr;301(1):95-102. [2] Jiang G, et al. J Med Chem. 2001 Feb 1;44(3):453-67.

参考

Molecular Formula	C₈₂H₁₀₃ClN₁₈O₁₆
Molecular Weight	1632.26
CAS No.	214766-78-6
Appearance	White Powder
Peptide Content (by %N)	≥80%
Single Impurity (by HPLC)	≤1.0%
Assay (By Anhydrous, Acetic Acid-free)	95.0~105.0%
MS	Consistent
Packing	plastic vial(dedicated for peptide packing) or glass vial, quantity according to customer's detail requirement.
Storage (From the date of receipt)	3 years-20°C powder
Shipping	Room temperature shipping(Stability testing shows this product can be shipped without any cooling measures.)