アロマターゼ

信号経路図

研究分野

  • 阻害剤の選択性比較
  • 溶解度
カタログ番号 製品カタログ 溶解度(25°C)
DMSO アルコール
S1235 Letrozole <1 mg/mL 57 mg/mL <1 mg/mL
S1188 Anastrozole <1 mg/mL 59 mg/mL 59 mg/mL
S1196 Exemestane <1 mg/mL 54 mg/mL 15 mg/mL
S2208 Formestane <1 mg/mL 61 mg/mL <1 mg/mL
S1672 Aminoglutethimide <1 mg/mL 20 mg/mL 7 mg/mL
製品コード 製品説明 文献中の使用例 お客様のフィードバック
S1235

Letrozole

Letrozole is a third generation inhibitor of aromatase with IC50 of 0.07-20 nM.

S1188

Anastrozole

Anastrozole inhibits the enzyme aromatase.

S1196

Exemestane

Exemestane was found to inhibit human placental aromatase with IC50 of 42 nM.

S2208

Formestane

Formestane is a second generation selective aromatase inhibitor with an IC50 of 80 nM.

S1672

Aminoglutethimide

Aminoglutethimide is aromatase inhibitor, also an P450scc inhibitor and blocks the conversion of cholesterol to pregnenolone.

製品コード 製品説明 文献中の使用例 お客様のフィードバック
S1235

Letrozole

Letrozole is a third generation inhibitor of aromatase with IC50 of 0.07-20 nM.

S1188

Anastrozole

Anastrozole inhibits the enzyme aromatase.

S1196

Exemestane

Exemestane was found to inhibit human placental aromatase with IC50 of 42 nM.

S2208

Formestane

Formestane is a second generation selective aromatase inhibitor with an IC50 of 80 nM.

S1672

Aminoglutethimide

Aminoglutethimide is aromatase inhibitor, also an P450scc inhibitor and blocks the conversion of cholesterol to pregnenolone.

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