アロマターゼ

信号経路図

研究分野

  • 阻害剤の選択性比較
  • 溶解度
カタログ番号 製品カタログ 溶解度(25°C)
DMSO アルコール
S1235 Letrozole <1 mg/mL 57 mg/mL <1 mg/mL
S1188 Anastrozole <1 mg/mL 59 mg/mL 59 mg/mL
S1196 Exemestane <1 mg/mL 54 mg/mL 15 mg/mL
S2208 Formestane <1 mg/mL 61 mg/mL <1 mg/mL
S1672 Aminoglutethimide <1 mg/mL 20 mg/mL 7 mg/mL
製品コード 製品説明 文献中の使用例 お客様のフィードバック
S1235

Letrozole

Letrozole is a third generation inhibitor of aromatase with IC50 of 0.07-20 nM.

S1188

Anastrozole

Anastrozole inhibits the enzyme aromatase.

S1196

Exemestane

Exemestane was found to inhibit human placental aromatase with IC50 of 42 nM.

S2208

Formestane

Formestane is a second generation selective aromatase inhibitor with an IC50 of 80 nM.

S1672

Aminoglutethimide

Aminoglutethimide is aromatase inhibitor, also an P450scc inhibitor and blocks the conversion of cholesterol to pregnenolone.

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