GRK antibodies| GRK antagonist | GRK inhibitor | GRK agonist

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Specific Compounds Quantities 96 or 384 well Plate Map Dry/solid or DMSO solution

抗体

製品コード	製品名称	製品説明	文献中Selleckの製品使用例
S8489	GSK180736A (GSK180736)	GSK180736A (GSK180736), developed as a Rho-associated, coiled-coil-containing protein kinase inhibitor, binds to GRK2(G protein-coupled receptor kinase 2) with logIC50 pf -6.6 (logIC50 -4.0 for GRK5 and >-3 for GRK1); ≥400-fold selective for GRK2 over both GRK1 and GRK5.	Cell Rep, 2023, 42(7):112812 Cancer Lett, 2022, 529:112-125
E2817	GRK5-IN-2	GRK5-IN-2 is a potent G-protein-coupled receptor kinase 5 (GRK5) inhibitor.
S6621	CCG215022	CCG215022 serves as a pan-G protein-coupled receptor kinases (GRKs) inhibitor with IC50 of 3.9 μM, 0.15 μM, 0.38 μM for GRK1, GRK2, GRK5, respectively.
S8489	GSK180736A (GSK180736)	GSK180736A (GSK180736), developed as a Rho-associated, coiled-coil-containing protein kinase inhibitor, binds to GRK2(G protein-coupled receptor kinase 2) with logIC50 pf -6.6 (logIC50 -4.0 for GRK5 and >-3 for GRK1); ≥400-fold selective for GRK2 over both GRK1 and GRK5.	Cell Rep, 2023, 42(7):112812 Cancer Lett, 2022, 529:112-125
E2817	GRK5-IN-2	GRK5-IN-2 is a potent G-protein-coupled receptor kinase 5 (GRK5) inhibitor.
S6621	CCG215022	CCG215022 serves as a pan-G protein-coupled receptor kinases (GRKs) inhibitor with IC50 of 3.9 μM, 0.15 μM, 0.38 μM for GRK1, GRK2, GRK5, respectively.

GRK

GRK製品

GRK阻害剤の選択性比較