phosphatase

  • 阻害剤の選択性比較
  • 溶解度
カタログ番号 製品カタログ 溶解度(25°C)
DMSO アルコール
S1949 Menadione <1 mg/mL 34 mg/mL 34 mg/mL
S1857 Etidronate 41 mg/mL <1 mg/mL <1 mg/mL
S1514 Cyclosporine <1 mg/mL 100 mg/mL 100 mg/mL
S4007 Pentamidine isethionate 100 mg/mL 100 mg/mL <1 mg/mL
S7437 Sal003 <1 mg/mL 93 mg/mL <1 mg/mL
S8278 SHP099 77 mg/mL 2 mg/mL <1 mg/mL
S8182 NSC87877 100 mg/mL 100 mg/mL <1 mg/mL
S4013 Sodium Monofluorophosphate 29 mg/mL <1 mg/mL <1 mg/mL
S7485 CCT007093 <1 mg/mL 1 mg/mL <1 mg/mL
S7537 LB-100 53 mg/mL <1 mg/mL <1 mg/mL
S7383 (-)-p-Bromotetramisole Oxalate 30 mg/mL 74 mg/mL <1 mg/mL
S7573 <1 mg/mL 92 mg/mL 92 mg/mL
製品コード 製品説明 文献中の使用例 お客様のフィードバック
S1949

Menadione

Menadione, a synthetic naphthoquinone without the isoprenoid side chain and biological activity, but can be converted to active vitamin K2, menaquinone, after alkylation in vivo.

S1857

Etidronate

Etidronate (Didronel) is a human protein tyrosine phosphatase inhibitor with IC50 of 0.2 μM.

S1514

Cyclosporine

Cyclosporine (Neoral) is an immunosuppressant drug.

S4007

Pentamidine isethionate

Pentamidine HClはPRLホスファターゼの阻害体、そのうえ、DNA、RNAとタンパク質の合成を禁止します。

S7437

Sal003

Sal003 is a potent and cell-permeable eIF-2α phosphatase inhibitor.

S8278

SHP099

S8182

NSC87877

S4013

Sodium Monofluorophosphate

Monofluorophosphateは競争的なピルビン酸塩キナーゼアルカリホスファターゼ阻害剤で、Ki がそれぞれ3.4 mM と 69 μMです。また、ホスホリラーゼ・ホスファターゼ を不可逆的に妨げます、 Ki が0.5 mMです。

S7485

CCT007093

CCT007093 is a potent PPM1D (WIP1) inhibitor with IC50 of 8.4 μM.

S7537

LB-100

LB-100 is a water soluble protein phosphatase 2A (PP2A) inhibitor. Phase 1.

S7383

(-)-p-Bromotetramisole Oxalate

(-)-p-Bromotetramisole Oxalate is a potent and non-specific alkaline phosphatase inhibitor.

製品コード 製品説明 文献中の使用例 お客様のフィードバック
S1949

Menadione

Menadione, a synthetic naphthoquinone without the isoprenoid side chain and biological activity, but can be converted to active vitamin K2, menaquinone, after alkylation in vivo.

S1857

Etidronate

Etidronate (Didronel) is a human protein tyrosine phosphatase inhibitor with IC50 of 0.2 μM.

S1514

Cyclosporine

Cyclosporine (Neoral) is an immunosuppressant drug.

S4007

Pentamidine isethionate

Pentamidine HClはPRLホスファターゼの阻害体、そのうえ、DNA、RNAとタンパク質の合成を禁止します。

S7437

Sal003

Sal003 is a potent and cell-permeable eIF-2α phosphatase inhibitor.

S8278

SHP099

S8182

NSC87877

S4013

Sodium Monofluorophosphate

Monofluorophosphateは競争的なピルビン酸塩キナーゼアルカリホスファターゼ阻害剤で、Ki がそれぞれ3.4 mM と 69 μMです。また、ホスホリラーゼ・ホスファターゼ を不可逆的に妨げます、 Ki が0.5 mMです。

S7485

CCT007093

CCT007093 is a potent PPM1D (WIP1) inhibitor with IC50 of 8.4 μM.

S7537

LB-100

LB-100 is a water soluble protein phosphatase 2A (PP2A) inhibitor. Phase 1.

S7383

(-)-p-Bromotetramisole Oxalate

(-)-p-Bromotetramisole Oxalate is a potent and non-specific alkaline phosphatase inhibitor.

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