AChR

信号経路図

研究分野

  • 阻害剤の選択性比較
  • 溶解度
カタログ番号 製品カタログ 溶解度(25°C)
DMSO アルコール
S2462 Donepezil HCl 5 mg/mL <1 mg/mL <1 mg/mL
S2547 Tiotropium Bromide hydrate <1 mg/mL 8 mg/mL <1 mg/mL
S2251 (-)-Huperzine A (HupA) <1 mg/mL 0.66 mg/mL <1 mg/mL
S2497 Pancuronium dibromide 100 mg/mL 100 mg/mL 100 mg/mL
S2550 Tolterodine tartrate 17 mg/mL 95 mg/mL 6 mg/mL
S4718 Acetylcholine iodide 54 mg/mL 54 mg/mL 54 mg/mL
S2240 Fesoterodine Fumarate 100 mg/mL 100 mg/mL 100 mg/mL
S3005 Paroxetine HCl 1 mg/mL 73 mg/mL 35 mg/mL
S2629 PNU-120596 <1 mg/mL 62 mg/mL 1 mg/mL
S1754 Oxybutynin <1 mg/mL 71 mg/mL 71 mg/mL
S2452 Amfebutamone (Bupropion) HCl <1 mg/mL 8 mg/mL <1 mg/mL
S3048 Solifenacin succinate 96 mg/mL 3 mg/mL 5 mg/mL
S1440 Varenicline Tartrate 72 mg/mL 1 mg/mL <1 mg/mL
S1339 Galanthamine HBr 36 mg/mL <1 mg/mL <1 mg/mL
S1405 Vecuronium Bromide 4 mg/mL 100 mg/mL 100 mg/mL
S1683 Ipratropium Bromide 83 mg/mL 83 mg/mL 83 mg/mL
S2549 Trospium chloride 86 mg/mL 41 mg/mL 42 mg/mL
S2130 Atropine sulfate monohydrate 139 mg/mL 139 mg/mL 139 mg/mL
S4031 Aclidinium Bromide <1 mg/mL 113 mg/mL <1 mg/mL
S1397 Rocuronium Bromide 122 mg/mL 122 mg/mL 122 mg/mL
S1978 Methscopolamine 67 mg/mL 79 mg/mL <1 mg/mL
S3047 Otilonium Bromide 113 mg/mL 113 mg/mL 113 mg/mL
S2508 Scopolamine HBr 76 mg/mL 76 mg/mL <1 mg/mL
S2455 Bethanechol chloride 39 mg/mL 39 mg/mL 39 mg/mL
S2471 Gallamine Triethiodide 100 mg/mL 100 mg/mL <1 mg/mL
S1608 Pyridostigmine Bromide 52 mg/mL 52 mg/mL 52 mg/mL
S2659 5-hydroxymethyl Tolterodine (PNU 200577, 5-HMT, 5-HM) <1 mg/mL 68 mg/mL 68 mg/mL
S2614 Arecoline HBr 47 mg/mL 47 mg/mL 10 mg/mL
S4231 Pilocarpine HCl 48 mg/mL 48 mg/mL 48 mg/mL
S2087 Rivastigmine Tartrate 80 mg/mL 42 mg/mL 80 mg/mL
S1929 Irsogladine <1 mg/mL 2 mg/mL <1 mg/mL
S2490 Neostigmine Bromide 60 mg/mL <1 mg/mL <1 mg/mL
S3144 Darifenacin HBr <1 mg/mL 100 mg/mL <1 mg/mL
S3202 Catharanthine <1 mg/mL 67 mg/mL 3 mg/mL
S4575 Pralidoxime (chloride) 34 mg/mL <1 mg/mL 1 mg/mL
S4014 Hyoscyamine <1 mg/mL 58 mg/mL 58 mg/mL
S4023 Procaine HCl 55 mg/mL 55 mg/mL <1 mg/mL
S4024 Homatropine Methylbromide 74 mg/mL 74 mg/mL 10 mg/mL
S4025 Homatropine Bromide 71 mg/mL 71 mg/mL <1 mg/mL
S4027 Flavoxate HCl 10 mg/mL 3 mg/mL <1 mg/mL
S4121 Succinylcholine Chloride Dihydrate 79 mg/mL 1 mg/mL <1 mg/mL
S2054 Orphenadrine Citrate <1 mg/mL 92 mg/mL <1 mg/mL
S4034 Diphemanil Methylsulfate 28 mg/mL 25 mg/mL <1 mg/mL
S4617 Dextromethorphan (hydrobromide hydrate) <1 mg/mL 74 mg/mL 74 mg/mL
S1832 Atracurium Besylate 33 mg/mL 100 mg/mL 100 mg/mL
S4143 Pentoxyverine Citrate 100 mg/mL 100 mg/mL 8 mg/mL
S4619 Itopride hydrochloride 78 mg/mL 78 mg/mL 38 mg/mL
S4422 Nitenpyram 54 mg/mL 54 mg/mL 54 mg/mL
S7366 LY2119620 <1 mg/mL 87 mg/mL 10 mg/mL
S4162 Benzethonium Chloride 90 mg/mL 90 mg/mL 90 mg/mL
S2287 Cytisine 38 mg/mL 38 mg/mL 38 mg/mL
S4171 Choline Chloride 28 mg/mL 28 mg/mL 28 mg/mL
S4069 Hexamethonium Dibromide 73 mg/mL <1 mg/mL <1 mg/mL
S4660 Glycopyrrolate 79 mg/mL 65 mg/mL 59 mg/mL
S4072 Decamethonium Bromide 84 mg/mL 34 mg/mL 25 mg/mL
S4505 Vinblastine sulfate <1 mg/mL 100 mg/mL <1 mg/mL
S3117 Oxybutynin chloride 4 mg/mL 79 mg/mL 79 mg/mL
S4542 Trihexyphenidyl hydrochloride <1 mg/mL 7 mg/mL 24 mg/mL
S2082 Adiphenine HCl 70 mg/mL 30 mg/mL 18 mg/mL
S4292 Diphenidol HCl 13 mg/mL 69 mg/mL 36 mg/mL
S1913 Tropicamide <1 mg/mL 57 mg/mL 57 mg/mL

亜型選択性的な製品

製品コード 製品説明 文献中の使用例 お客様のフィードバック
S2462

Donepezil HCl

Donepezil HCl はbAChEとhAChEのための8.12nMと11.6nMのIC50によるアセチルコリンエステラーゼ(AChE)の特定で強力な阻害剤です。

S2251

(-)-Huperzine A (HupA)

(-)-Huperzine A (HupA)は アセチルコリンエステラーゼ(AChE)の強力で、非常に特定で、可逆的な阻害剤で、Ki が 7 nMです。

S2452

Amfebutamone (Bupropion) HCl

Amfebutamone (Bupropion) HCl is a selective norepinephrine-dopamine reuptake inhibitor with IC50 of 6.5 and 3.4μM for the reuptake of dopamine and norepinephrine, respectively

S1339

Galanthamine HBr

Galanthamine HBrは、IC50が14nMによりある長時間作用性のアセチルコリンエステラーゼ(AChE)阻害剤です。

S4031

Aclidinium Bromide

Aclidinium Bromideは人間のムスカリン性 AChR のM1、M2、M3、M4とM5をバインド、Ki がそれぞれ 0.1 nM、 0.14 nM、 0.14 nM、 0.21 nM と 0.16 nMです。

S1397

Rocuronium Bromide

Rocuronium Bromide is an aminosteroid non-depolarizing neuromuscular blocker or muscle relaxant.

S3047

Otilonium Bromide

Otilonium bromide is an antimuscarinic.

S2471

Gallamine Triethiodide

Gallamine Triethiodide is a cholinergic receptor blocker with an IC50 of 68.0 ± 8.4 μM.

S1608

Pyridostigmine Bromide

Pyridostigmine Bromide is a parasympathomimetic and a reversible cholinesterase inhibitor.

S2087

Rivastigmine Tartrate

Rivastigmine Tartrate, a cholinesterase inhibitor with IC50 of 5.5 μM, ues as a parasympathomimetic or cholinergic agent for the treatment of mild to moderate Alzheimer disease.

S1929

Irsogladine

Irsogladine is an anti-gastric ulcer agent that facilitates gap-junctional intercellular communication through M1 muscarininc acetylcholine receptor binding.

S2490

Neostigmine Bromide

Neostigmine Bromide is a reversible acetylcholinesterase inhibitor.

S3202

Catharanthine

Catharanthine inhibits nicotinic receptor mediated diaphragm contractions with IC50 of 59.6 μM

S4014

Hyoscyamine

Hyoscyamine は、AChR 阻害剤で、IC50 が 7.5 nMです。

S4023

Procaine HCl

Procaine HCl is an inhibitor of sodium channel, NMDA receptor and nicotinic acetylcholine receptors with IC50 of 60 μM, 0.296 mM and 45.5 μM, which is also an inhibitor of 5-HT3 with KD of 1.7 μM.

S1832

Atracurium Besylate

Atracurium Besylate is a neuromuscular blocking agent with ED95 of 0.2 mg/kg.

S4619

Itopride hydrochloride

S4162

Benzethonium Chloride

Benzethonium chloride is a potent inhibitor of neuronal nicotinic acetylcholine receptors (nAChRs), it inhibits α4β2 nAChRs and α7 nAChRs with IC50of 49 nM and 122 nM, respectively.

S4505

Vinblastine sulfate

Vinblastine sulfateはマイクロチューブ形成とnAChR活性を抑制して、無細胞試験でIC50値が8.9μMになりますが、いくつかの種類癌症の治療に使用されます。

S4687

Rivastigmine

Rivastigmineは1種のコリンエステラーゼ(cholinesterase)阻害剤(IC50:5.5 μM)で、アセチルコリンエステラーゼ(acetylcholinesterase)((IC50 : 4.15 µM) )とブチリルコリンエステラーゼ(butyrylcholinesterase)((IC50 : 37 nM)を抑制します。

S4542

Trihexyphenidyl hydrochloride

S2082

Adiphenine HCl

Adiphenine is a nicotinic receptor inhibitor with IC50 of 15 µM, used as an antispasmodic drug.

S2547

Tiotropium Bromide hydrate

Tiotropium Bromide hydrate is a monohydrate of tiotropium bromide (Spiriva; Tiova; BA 679BR; tiopropium) that is an anticholinergic and bronchodilator and a muscarinic receptor antagonist.

S2497

Pancuronium dibromide

Pancuronium dibromide is a competitive acetylcholine antagonist with an IC50 of 5.5 nM.

S2550

Tolterodine tartrate

Tolterodine tartrate is a tartrate salt of tolterodine that is a competitive muscarinic receptor antagonist.

S2240

Fesoterodine Fumarate

Fesoterodine Fumarate is an antimuscarinic agent and is rapidly de-esterified to its active metabolite 5-hydroxymethyl tolterodine that is a muscarinic receptor antagonist.

S1754

Oxybutynin

Oxybutynin is an anticholinergic medication used to relieve urinary and bladder difficulties.

S3048

Solifenacin succinate

Solifenacin succinate is a urinary antispasmodic of the antimuscarinic class.

S1683

Ipratropium Bromide

Ipratropium bromide is a muscarinic antagonist, bronchodilator, N-Isopropyl salt of atropine.

S2549

Trospium chloride

Trospium chloride is a competitive muscarinic cholinergic receptor antagonist.

S2130

Atropine sulfate monohydrate

Atropine is a competitive muscarinic acetylcholine receptor antagonist with an IC50 of 2.5 nM.

S1978

Methscopolamine

Methscopolamine is a muscarinic acetylcholine receptor blocker.

S2508

Scopolamine HBr

Scopolamine HBr is a competitive muscarinic acetylcholine receptor with an IC50 of 55.3 nM.

S2659

5-hydroxymethyl Tolterodine (PNU 200577, 5-HMT, 5-HM)

5-hydroxymethyl Tolterodine (PNU 200577, 5-HMT, 5-HM) is a potent muscarinic receptor antagonist with a Kb and a pA2 of 0.84 nM and 9.14, respectively.

S3144

Darifenacin HBr

Darifenacin HBr is a selective M3 muscarinic receptor antagonist with pKi of 8.9.

S4024

Homatropine Methylbromide

Homatropine Methylbromideは、ムスカリンAChR敵対者、WKY-EとSHR-Eを妨げます。IC50 がそれぞれ 162.5 nM と 170.3 nMです。

S4025

Homatropine Bromide

Homatropine Bromideは、ムスカリンAChR敵対者、WKY-EとSHR-Eを妨げます。IC50 がそれぞれ 162.5 nM と 170.3 nMです。

S4027

Flavoxate HCl

Flavoxate HClは、ムスカリン性AChRの拮抗剤で、IC50 が12.2 μMです。

S2054

Orphenadrine Citrate

Orphenadrine citrate is a skeletal muscle relaxant, it acts in the central nervous system to produce its muscle relaxant effects.

S4034

Diphemanil Methylsulfate

Diphemanil Methylsulfateはアンモニウム抗コリン作用薬で、それはムスカリン性アセチルコリン受容体に結合します。(mAchR)

S4143

Pentoxyverine Citrate

Pentoxyverine (Carbetapentane) Citrateは、鎮咳性一般に風邪のような病気を伴う咳のために使われます。

S4069

Hexamethonium Dibromide

Hexamethonium Dibromideは AChR の神経型ニコチン性選択的アンタゴニストです。

S4660

Glycopyrrolate

Glycopyrrolateは1種のムスカリン性(muscarinic)の拮抗剤です。胃腸管の疾病に於いて、Glycopyrrolateは鎮痙薬として使用されます。

S3117

Oxybutynin chloride

Oxybutynin chloride is an anticholinergic medication used to relieve urinary and bladder difficulties.

S4292

Diphenidol HCl

Diphenidol HCl is a potent antagonist of muscarinic M2 and M3 receptor with pKb of 6.72 and 7.02, respectively, used in the treatment of vomiting and vertigo.

S1913

Tropicamide

Tropicamide is an anticholinergic and a muscarinic receptor subtype M4-preferring antagonist with IC50 of 8.0 nM.

S2629

PNU-120596

PNU-120596はα7つの<夕食をとります>*<の216nMのEC50によるα7つのnAChRの陽アロステリックモジュレーターです/>を表しているSH-EP1細胞をすすってください。

S4718

Acetylcholine iodide

S1440

Varenicline Tartrate

Varenicline Tartrate is a prescription medication used to treat smoking addiction.

S2455

Bethanechol chloride

Bethanechol chloride is a selective muscarinic receptor agonist without any effect on nicotinic receptors.

S2614

Arecoline HBr

Arecoline is a muscarinic acetylcholine receptor agonist.

S4231

Pilocarpine HCl

Pilocarpine HCl is a nonselective muscarinic acetylcholine receptor agonist used to produce an experimental model of epilepsy.

S4121

Succinylcholine Chloride Dihydrate

Succinylcholine Chloride Dihydrate is a nicotinic AChR agonist and also acts as a depolarizing neuromuscular blocker.

S4422

Nitenpyram

Nitenpyram is a nicotinic acetylcholine receptor (AchR) agonist, used as veterinary medicine to treat parasites of livestock and pets.

S7366

LY2119620

LY2119620 is a specific, and allosteric agonist of human M2 and M4 muscarinic acetylcholine receptors.

S2287

Cytisine

Cytisine is a nicotinic acetylcholine receptor agonist.

S4171

Choline Chloride

Choline chlorideは、動物用飼料添加剤として使用される第四級アンモニウム塩です。

S4072

Decamethonium Bromide

Decamethonium Bromideはニコチン性 AChRの部分アゴニストおよび運動支配のブロッキング剤です。

S1405

Vecuronium Bromide

Vecuronium Bromide is a muscle relaxant in the category of non-depolarizing blocking agents.

S4617

Dextromethorphan (hydrobromide hydrate)

S4575

Pralidoxime (chloride)

製品コード 製品説明 文献中の使用例 お客様のフィードバック
S2462

Donepezil HCl

Donepezil HCl はbAChEとhAChEのための8.12nMと11.6nMのIC50によるアセチルコリンエステラーゼ(AChE)の特定で強力な阻害剤です。

S2251

(-)-Huperzine A (HupA)

(-)-Huperzine A (HupA)は アセチルコリンエステラーゼ(AChE)の強力で、非常に特定で、可逆的な阻害剤で、Ki が 7 nMです。

S2452

Amfebutamone (Bupropion) HCl

Amfebutamone (Bupropion) HCl is a selective norepinephrine-dopamine reuptake inhibitor with IC50 of 6.5 and 3.4μM for the reuptake of dopamine and norepinephrine, respectively

S1339

Galanthamine HBr

Galanthamine HBrは、IC50が14nMによりある長時間作用性のアセチルコリンエステラーゼ(AChE)阻害剤です。

S4031

Aclidinium Bromide

Aclidinium Bromideは人間のムスカリン性 AChR のM1、M2、M3、M4とM5をバインド、Ki がそれぞれ 0.1 nM、 0.14 nM、 0.14 nM、 0.21 nM と 0.16 nMです。

S1397

Rocuronium Bromide

Rocuronium Bromide is an aminosteroid non-depolarizing neuromuscular blocker or muscle relaxant.

S3047

Otilonium Bromide

Otilonium bromide is an antimuscarinic.

S2471

Gallamine Triethiodide

Gallamine Triethiodide is a cholinergic receptor blocker with an IC50 of 68.0 ± 8.4 μM.

S1608

Pyridostigmine Bromide

Pyridostigmine Bromide is a parasympathomimetic and a reversible cholinesterase inhibitor.

S2087

Rivastigmine Tartrate

Rivastigmine Tartrate, a cholinesterase inhibitor with IC50 of 5.5 μM, ues as a parasympathomimetic or cholinergic agent for the treatment of mild to moderate Alzheimer disease.

S1929

Irsogladine

Irsogladine is an anti-gastric ulcer agent that facilitates gap-junctional intercellular communication through M1 muscarininc acetylcholine receptor binding.

S2490

Neostigmine Bromide

Neostigmine Bromide is a reversible acetylcholinesterase inhibitor.

S3202

Catharanthine

Catharanthine inhibits nicotinic receptor mediated diaphragm contractions with IC50 of 59.6 μM

S4014

Hyoscyamine

Hyoscyamine は、AChR 阻害剤で、IC50 が 7.5 nMです。

S4023

Procaine HCl

Procaine HCl is an inhibitor of sodium channel, NMDA receptor and nicotinic acetylcholine receptors with IC50 of 60 μM, 0.296 mM and 45.5 μM, which is also an inhibitor of 5-HT3 with KD of 1.7 μM.

S1832

Atracurium Besylate

Atracurium Besylate is a neuromuscular blocking agent with ED95 of 0.2 mg/kg.

S4619

Itopride hydrochloride

S4162

Benzethonium Chloride

Benzethonium chloride is a potent inhibitor of neuronal nicotinic acetylcholine receptors (nAChRs), it inhibits α4β2 nAChRs and α7 nAChRs with IC50of 49 nM and 122 nM, respectively.

S4505

Vinblastine sulfate

Vinblastine sulfateはマイクロチューブ形成とnAChR活性を抑制して、無細胞試験でIC50値が8.9μMになりますが、いくつかの種類癌症の治療に使用されます。

S4687

Rivastigmine

Rivastigmineは1種のコリンエステラーゼ(cholinesterase)阻害剤(IC50:5.5 μM)で、アセチルコリンエステラーゼ(acetylcholinesterase)((IC50 : 4.15 µM) )とブチリルコリンエステラーゼ(butyrylcholinesterase)((IC50 : 37 nM)を抑制します。

S4542

Trihexyphenidyl hydrochloride

S2082

Adiphenine HCl

Adiphenine is a nicotinic receptor inhibitor with IC50 of 15 µM, used as an antispasmodic drug.

製品コード 製品説明 文献中の使用例 お客様のフィードバック
S4575

Pralidoxime (chloride)

製品コード 製品説明 文献中の使用例 お客様のフィードバック
S2547

Tiotropium Bromide hydrate

Tiotropium Bromide hydrate is a monohydrate of tiotropium bromide (Spiriva; Tiova; BA 679BR; tiopropium) that is an anticholinergic and bronchodilator and a muscarinic receptor antagonist.

S2497

Pancuronium dibromide

Pancuronium dibromide is a competitive acetylcholine antagonist with an IC50 of 5.5 nM.

2014, (84):e51271

S2550

Tolterodine tartrate

Tolterodine tartrate is a tartrate salt of tolterodine that is a competitive muscarinic receptor antagonist.

S2240

Fesoterodine Fumarate

Fesoterodine Fumarate is an antimuscarinic agent and is rapidly de-esterified to its active metabolite 5-hydroxymethyl tolterodine that is a muscarinic receptor antagonist.

S1754

Oxybutynin

Oxybutynin is an anticholinergic medication used to relieve urinary and bladder difficulties.

S3048

Solifenacin succinate

Solifenacin succinate is a urinary antispasmodic of the antimuscarinic class.

S1683

Ipratropium Bromide

Ipratropium bromide is a muscarinic antagonist, bronchodilator, N-Isopropyl salt of atropine.

S2549

Trospium chloride

Trospium chloride is a competitive muscarinic cholinergic receptor antagonist.

S2130

Atropine sulfate monohydrate

Atropine is a competitive muscarinic acetylcholine receptor antagonist with an IC50 of 2.5 nM.

S1978

Methscopolamine

Methscopolamine is a muscarinic acetylcholine receptor blocker.

S2508

Scopolamine HBr

Scopolamine HBr is a competitive muscarinic acetylcholine receptor with an IC50 of 55.3 nM.

S2659

5-hydroxymethyl Tolterodine (PNU 200577, 5-HMT, 5-HM)

5-hydroxymethyl Tolterodine (PNU 200577, 5-HMT, 5-HM) is a potent muscarinic receptor antagonist with a Kb and a pA2 of 0.84 nM and 9.14, respectively.

S3144

Darifenacin HBr

Darifenacin HBr is a selective M3 muscarinic receptor antagonist with pKi of 8.9.

S4024

Homatropine Methylbromide

Homatropine Methylbromideは、ムスカリンAChR敵対者、WKY-EとSHR-Eを妨げます。IC50 がそれぞれ 162.5 nM と 170.3 nMです。

S4025

Homatropine Bromide

Homatropine Bromideは、ムスカリンAChR敵対者、WKY-EとSHR-Eを妨げます。IC50 がそれぞれ 162.5 nM と 170.3 nMです。

S4027

Flavoxate HCl

Flavoxate HClは、ムスカリン性AChRの拮抗剤で、IC50 が12.2 μMです。

S2054

Orphenadrine Citrate

Orphenadrine citrate is a skeletal muscle relaxant, it acts in the central nervous system to produce its muscle relaxant effects.

S4034

Diphemanil Methylsulfate

Diphemanil Methylsulfateはアンモニウム抗コリン作用薬で、それはムスカリン性アセチルコリン受容体に結合します。(mAchR)

S4143

Pentoxyverine Citrate

Pentoxyverine (Carbetapentane) Citrateは、鎮咳性一般に風邪のような病気を伴う咳のために使われます。

S4069

Hexamethonium Dibromide

Hexamethonium Dibromideは AChR の神経型ニコチン性選択的アンタゴニストです。

S4660

Glycopyrrolate

Glycopyrrolateは1種のムスカリン性(muscarinic)の拮抗剤です。胃腸管の疾病に於いて、Glycopyrrolateは鎮痙薬として使用されます。

S3117

Oxybutynin chloride

Oxybutynin chloride is an anticholinergic medication used to relieve urinary and bladder difficulties.

S4292

Diphenidol HCl

Diphenidol HCl is a potent antagonist of muscarinic M2 and M3 receptor with pKb of 6.72 and 7.02, respectively, used in the treatment of vomiting and vertigo.

S1913

Tropicamide

Tropicamide is an anticholinergic and a muscarinic receptor subtype M4-preferring antagonist with IC50 of 8.0 nM.

製品コード 製品説明 文献中の使用例 お客様のフィードバック
S4718

Acetylcholine iodide

S1440

Varenicline Tartrate

Varenicline Tartrate is a prescription medication used to treat smoking addiction.

S2455

Bethanechol chloride

Bethanechol chloride is a selective muscarinic receptor agonist without any effect on nicotinic receptors.

S2614

Arecoline HBr

Arecoline is a muscarinic acetylcholine receptor agonist.

2015, 33(6):2753-60

S4231

Pilocarpine HCl

Pilocarpine HCl is a nonselective muscarinic acetylcholine receptor agonist used to produce an experimental model of epilepsy.

S4121

Succinylcholine Chloride Dihydrate

Succinylcholine Chloride Dihydrate is a nicotinic AChR agonist and also acts as a depolarizing neuromuscular blocker.

S4422

Nitenpyram

Nitenpyram is a nicotinic acetylcholine receptor (AchR) agonist, used as veterinary medicine to treat parasites of livestock and pets.

S7366

LY2119620

LY2119620 is a specific, and allosteric agonist of human M2 and M4 muscarinic acetylcholine receptors.

S2287

Cytisine

Cytisine is a nicotinic acetylcholine receptor agonist.

S4171

Choline Chloride

Choline chlorideは、動物用飼料添加剤として使用される第四級アンモニウム塩です。

S4072

Decamethonium Bromide

Decamethonium Bromideはニコチン性 AChRの部分アゴニストおよび運動支配のブロッキング剤です。

製品コード 製品説明 文献中の使用例 お客様のフィードバック
S2629

PNU-120596

PNU-120596はα7つの<夕食をとります>*<の216nMのEC50によるα7つのnAChRの陽アロステリックモジュレーターです/>を表しているSH-EP1細胞をすすってください。

2016, 10.1007/s12035-016-9796-3

2013, 8(8): e73581

2017, 54(3):2045-2059

製品コード 製品説明 文献中の使用例 お客様のフィードバック
S1405

Vecuronium Bromide

Vecuronium Bromide is a muscle relaxant in the category of non-depolarizing blocking agents.

S4617

Dextromethorphan (hydrobromide hydrate)