Lipase

阻害剤の選択性比較

カタログ番号 製品カタログ 溶解度(25°C)
DMSO アルコール
S1629 Orlistat <1 mg/mL 99 mg/mL 99 mg/mL
S4904 JZL184 <1 mg/mL 100 mg/mL <1 mg/mL
S7364 Atglistatin <1 mg/mL 56 mg/mL 4 mg/mL
S7457 XEN445 <1 mg/mL 80 mg/mL 34 mg/mL
S9234 Schaftoside -1 mg/mL 100 mg/mL -1 mg/mL
S8823 ABX-1431 <1 mg/mL 100 mg/mL 100 mg/mL
S2365 Tanshinone IIA <1 mg/mL 5 mg/mL <1 mg/mL
S4930 Cetilistat <1 mg/mL 3 mg/mL 8 mg/mL
S4825 Pancreatin <1 mg/mL 0.01 mg/mL <1 mg/mL

Lipase製品

新Lipase製品
製品コード 製品説明 文献中Selleckの製品使用例 お客様のフィードバック
S1629

Orlistat

Orlistat is a general lipase inhibitor with IC50 of 122 ng/ml for PL from human duodenal juice.

S4904

JZL184

JZL 184 is the first selective inhibitor of monoacylglycerol lipase (MAGL) with IC50 of 8 nM.

S7364

Atglistatin

Atglistatin is a highly potent, and selective inhibitor of adipose triglyceride lipase (ATGL) with IC50 of 0.7 μM, high selectivity over other key metabolic lipases.

S7457

XEN445

XEN445 is a potent and selective endothelial lipase inhibitor with IC50 of 0.237 μM.

S9234

Schaftoside

Schaftoside, a bioactive compound found in the Herba Desmodii Styracifolii, exhibits pancreatic lipase inhibitory activity.

S8823

ABX-1431

ABX-1431 is a highly potent, selective, and CNS-penetrant Monoacylglycerol lipase (MGLL) inhibitor with IC50 values of 14 nM and 27 nM for hMGLL and mMGLL respectively.

S2365

Tanshinone IIA

Tanshinone IIA(Tanshinone B) is the most abundant diterpene quinone in Danshen, Salviae miltiorrhizae Radix, a widely prescribed traditional herbal medicine that is used to treat cardiovascular and inflammatory diseases; A natural monoacylglycerol lipase inhibitor.

S4930

Cetilistat

Cetilistat is a novel highly lipophilic benzoxazinone that inhibits gastrointestinal and pancreatic lipases. It shows a good safety and tolerability profile in vivo

S4825

Pancreatin

Pancreatic enzymes also known as pancrelipase and pancreatin, are commercial mixtures of amylase, lipase, and protease. They are used to treat malabsorption syndrome due to pancreatic problems.

製品コード 製品説明 文献中Selleckの製品使用例 お客様のフィードバック
S1629

Orlistat

Orlistat is a general lipase inhibitor with IC50 of 122 ng/ml for PL from human duodenal juice.

S4904

JZL184

JZL 184 is the first selective inhibitor of monoacylglycerol lipase (MAGL) with IC50 of 8 nM.

S7364

Atglistatin

Atglistatin is a highly potent, and selective inhibitor of adipose triglyceride lipase (ATGL) with IC50 of 0.7 μM, high selectivity over other key metabolic lipases.

S7457

XEN445

XEN445 is a potent and selective endothelial lipase inhibitor with IC50 of 0.237 μM.

S9234

Schaftoside

Schaftoside, a bioactive compound found in the Herba Desmodii Styracifolii, exhibits pancreatic lipase inhibitory activity.

S8823

ABX-1431

ABX-1431 is a highly potent, selective, and CNS-penetrant Monoacylglycerol lipase (MGLL) inhibitor with IC50 values of 14 nM and 27 nM for hMGLL and mMGLL respectively.

S2365

Tanshinone IIA

Tanshinone IIA(Tanshinone B) is the most abundant diterpene quinone in Danshen, Salviae miltiorrhizae Radix, a widely prescribed traditional herbal medicine that is used to treat cardiovascular and inflammatory diseases; A natural monoacylglycerol lipase inhibitor.

S4930

Cetilistat

Cetilistat is a novel highly lipophilic benzoxazinone that inhibits gastrointestinal and pancreatic lipases. It shows a good safety and tolerability profile in vivo

製品コード 製品説明 文献中Selleckの製品使用例 お客様のフィードバック
S4825

Pancreatin

Pancreatic enzymes also known as pancrelipase and pancreatin, are commercial mixtures of amylase, lipase, and protease. They are used to treat malabsorption syndrome due to pancreatic problems.

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