GPCR Compound Library

目录号 L2200

Selleck GPCR Small Molecule Compound Library contains various small molecules targeting G protein coupled receptors with biological activity.

サイズ 価格(税別)  
予めDMSOまたは水に溶解しています
1226800
1799500
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GPCR Compound Library内容

Download theGPCR Compound Library - SDF
Download theGPCR Compound Library - XLSX

Selleckの分子ライブラリーが使用されている文献(42)

製品特性＆メリット

・Gタンパク質共役受容体をターゲットとした722種類の化合物ライブラリーです。HTS（High Throughput Screening） およびHCS（High Content Screening）に使用できます。

・ライブラリーの化合物は全て生物活性と薬理活性を有しています。

・オーファンGPCR（Orphan GPCR）は機能未知なため、弊社のGPCR化合物ライブラリーを使用することで機能未知のGPCRsを選別し、新たなGPCR標的薬を見出す可能性があります。

・GPCR化合物ライブラリーは様々な受容体（5-HT受容体、ドーパミン受容体、オピオイド受容体、アドレナリン受容体、カンナビノイド受容体、代謝型グルタミン酸受容体、エンドセリン受容体など）を標的としています。

・構造的に多様で、薬効および細胞透過性が確認されています。

・詳しい構造説明と、お客様からのレビューなど豊富な情報があります。

・NMRとHPLC検査で製品の高純度を保証しています。

製品詳細情報

調合： 658 compounds pre-dissolved in 10mM DMSO, 40 compounds pre-dissolved in 10mM water, 20 compounds pre-dissolved in 2mM DMSO and 4 compounds pre-dissolved in 2mM water
ケース： 96/384 Well Format Sample Storage Tube With Screw Cap and Optional 2D Barcode
安定性： in DMSO
in DMSO
出荷方式： ブルーアイス物流
包装： 不活性ガス（Inert gas）

GPCR Compound Library组成

HTS パートナ

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