Macrocyclic Compound Library

目录号 L7300

A unique collection of 104 macrocyclic compounds used for high throughput screening(HTS) and high content screening(HCS).

サイズ

価格(税別)

予めDMSOまたは水に溶解しています
100uL/well (2mM or 10mM solution)	510200

最寄りの販売代理店を探す

東京
北海道
東北
北関東
南関東
東海
北信越
近畿
中国
四国
九州

お探しのディーラーが見当たらない場合は直接こちらのメールアドレスまでお問い合わせください：[email protected]

具体的な在庫状況を確認してください。代表番号: 03-5615-9297 | 電子メール：[email protected]

セレックの化合物ライブラリーはCOVID19研究に貢献しています

(日本)国立感染症研究所はセレックのFDA承認化合物を用いてスクリニーング実験を行い、研究から僅か3ヶ月以内にCOVID19
の治療薬候補を見出しました。本研究成果はBioRxivにて発表されました。doi: 10.1101/2020.04.14.039925。

本研究成果はテレビニュース等での報道も行われました

お気に入りの分子或いは調達サービスにより、分子ライブラリーをカスタマイズします。
お客様自身のニーズを満たすために、弊社の製品を数量、状態（乾燥状態/固体或いはDMSO）等で選択できます。

Macrocyclic Compound Library内容

Download theMacrocyclic Compound Library - SDF

Download theMacrocyclic Compound Library - XLSX

Download the Compound Library Usage Instructions- PDF

Selleckの分子ライブラリーが使用されている文献(73)

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Genome Biol,2019,20(1):253

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Sci Adv,2019,5(6):eaav9784

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Cell Rep,2019,5;26(6):1544-1556.e8.

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Neuropsychopharmacology,2019,10.1038/s41386-018-0266-7

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Cancers (Basel),2019,30;11(2):156.

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Breast Cancer Res,2019,21(1):37

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Neurobiol Aging,2019,76:24-34

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Cancer Gene Ther,2019,10.1038/s41417-019-0127-5

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Stem Cells Int,2019,2019:3435901

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Cancer Manag Res,2019,11:8391-8405

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Breast Cancer Res Treat,2019,10.1007/s10549-019-05504-5

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Acta Pharmacol Sin,2019,10.1038/s41401-019-0246-4

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bioRxiv,2019,doi:10.1101/748129

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Nat Commun,2018,9(1):1655

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Selleck化合物ライブラリー使用例

肝癌研究におけるGPCR Compound Libraryの使用例（当文献はNature (IF=43)に掲載され、研究期間は約15ヶ月です）：
Nature.2019;574(7777):268-272
大腸癌研究におけるKinase Inhibitor Library の使用例（当文献はNature Communications (IF=11)に掲載され、研究期間は約8ヶ月です）：
Nat Commun. 2019 16;10(1):2197
抗ウイルス研究におけるFDA-approved Drug Libraryの使用例（当文献はCell Research (IF=17)に掲載され、研究期間は約13ヶ月です）：
Cell Res. 2019;29(9):739-753
代謝研究におけるFDA-approved Drug Library使用例（当文献はMovement Disorders (IF=8)に掲載され、研究期間は約10ヶ月です）：
Mov Disord. 2019;34(3):323-334
白血病研究におけるEpigenetics Compound Libraryの使用例（当文献は Blood (IF=16)に掲載され、研究期間は約16ヶ月です）：
Blood. 2019 17;134(16):1323-1336
癌免疫研究におけるInhibitor Libraryの使用例（当文献はCancer Immunol Res (IF=8.6)に掲載され、研究期間は約12ヶ月です）：
Cancer Immunol Res.2017;5(9):790-803

製品特性＆メリット

•Macrocycles are often described as molecules and ions containing twelve or more membered ring. Macrocycles often bind ions and facilitate ion transport across hydrophobic membranes and solvents.Macrocycles are often bioactive and could be useful for drug delivery

•A unique collection of 104 macrocyclic compounds used for high throughput screening(HTS) and high content screening(HCS)

•Some compounds have been approved by the FDA

•Structurally diverse,medicinally active,and cell permeable

•Rich documentation with structure and bioactivity information

•NMR and HPLC validated to ensure high purity

製品詳細情報

調合：	84 compounds pre-dissolved in 10mM DMSO, 19 compounds pre-dissolved in 10mM water and 1 compounds pre-dissolved in 2mM water
ケース：	96/384 Well Format Sample Storage Tube With Screw Cap and Optional 2D Barcode
安定性：	12 months -20°Cin DMSO
安定性：	24 months -80°Cin DMSO
出荷方式：	ブルーアイス物流
包装：	不活性ガス（Inert gas）

Macrocyclic Compound Library组成

HTS パートナ

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研究分野別

製品類型