| 製品コード |
製品名 |
製品説明 |
| S5079 |
Sitagliptin |
Sitagliptin (MK-0431) is an oral and highly selective DPP-4 inhibitor with an IC50 of 18 nM. It is used for the treatment of type 2 diabetes. |
| S5066 |
Pramipexole dihydrochloride |
Pramipexole dihydrochloride (SND919) is a dopamine agonist of the non-ergoline class indicated for treating Parkinson's disease (PD) and restless legs syndrome (RLS) with Ki values of 3.9 nM, 2.2 nM, 0.5 nM and 5.1 nM for D2S receptor, D2L receptor, D3 receptor and D4 receptor. |
| S5244 |
Zoledronic acid monohydrate |
Zoledronic acid (Zoledronate, CGP-4244) monohydrate, a nitrogen-containing bisphosphonate, is a potent osteoclast inhibitor which induces apoptosis in osteoclasts by inhibiting enzymes of the mevalonate pathway and preventing the isoprenylation of small GTP-binding proteins such as Ras and Rho. |
| S5527 |
Salmeterol |
Salmeterol (Astmerole, GR-33343X, SN408D) is a long-acting beta2-adrenergic receptor agonist with Ki value of 1.5 nM for WT β2AR and shows very high selectivity for the WT β2AR(β1Ki/β2Ki ratio of approximately 1500). |
| S5248 |
Apatinib |
Apatinib is a potent inhibitor of the VEGF signaling pathway with IC50 values of 1 nM, 13 nM, 429 nM and 530 nM for VEGFR-2, Ret (c-Ret), c-Kit and c-Src, respectively. Apatinib induces both autophagy and apoptosis. |
| S5480 |
Clidinium Bromide |
Clidinium Bromide is an anticholinergic drug. |
| S5484 |
Rimantadine Hydrochloride |
Rimantadine is an RNA synthesis inhibitor that is used as an antiviral agent in the prophylaxis and treatment of influenza. It works by inhibiting a viral protein called M2, which normally mediates the transport of acid ions across the influenza virion shell. |
| S5490 |
Disopyramide |
Disopyramide is a class IA antiarrhythmic drug which acts via blockade of sodium channels depressing phase 0 of the action potential. Disopyramide possesses significant negative inotropic, anticholinergic effects and enhances AV nodal conduction. |
| S5215 |
Abacavir |
Abacavir (ABC) is a powerful nucleoside analog reverse transcriptase inhibitor (NRTI) used to treat HIV and AIDS. |
| S5250 |
Darunavir |
Darunavir (TMC114) is a nonpeptidic HIV protease inhibitor, used to treat HIV infection. |
| S5098 |
Gefitinib hydrochloride |
Gefitinib (ZD1839) is an EGFR inhibitor with IC50s of 15.5 nM and 823.3 nM for WT EGFR and EGFR (858R/T790M), respectively. |
| S4996 |
Tavaborole (AN-2690) |
Tavaborole (AN-2690) is a boron-containing small molecule with broad spectrum antifungal activity. |
| S5481 |
Molindone hydrochloride |
Molindone hydrochloride is the hydrochloride salt form of molindone, a conventional antipsychotic used in the therapy of schizophrenia. It is a dopamine D2/D5 receptor antagonist. |
| S5492 |
Econazole |
Econazole is a broad spectrum antimycotic with some action against Gram positive bacteria. |
| S5499 |
Amantadine |
Amantadine (1-Adamantanamine, 1-Adamantylamine, 1-Aminoadamantane) is an antiviral that is used in the prophylactic or symptomatic treatment of influenza A. It is an M2 inhibitor which blocks the ion channel formed by the M2 protein that spans the viral membrane. |
| S5320 |
Octinoxate |
Octinoxate (Octyl methoxycinnamate, ethylhexyl methoxycinnamate) is a cinnamate ester and common ingredient in sunscreen and other skin care products to minimize DNA photodamage. |
| S5296 |
Cephradine monohydrate |
Cefradine is a beta-lactam, first-generation cephalosporin antibiotic with bactericidal activity. |
| S5298 |
Amoxicillin trihydrate |
Amoxicillin (Amoxil, Amoxipen, Moxaline) is a broad-spectrum, semisynthetic aminopenicillin antibiotic with bactericidal activity. |
| S5497 |
Iopanoic acid |
Iopanoic acid (Acidum iopanoicum, Iodopanoic acid) is an iodine-containing radiocontrast medium used in cholecystography. |
| S5515 |
Penicillin G Procaine |
Procaine benzylpenicillin (Procaine benzylpenicillin), also known as Procaine benzylpenicillin, is an antibiotic useful for the treatment of a number of bacterial infections. |
