FDA-approved & Passed Phase I Drug Library

目录号 L3800

A unique collection of 2880 drugs that are marketed around the world or that have passed phase 1 clinical trials for high throughput screening (HTS) and high content screening (HCS).

サイズ 価格(税別)  
予めDMSOまたは水に溶解しています
3191300
5104900
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セレックの化合物ライブラリーはCOVID19研究に貢献しています

(日本)国立感染症研究所はセレックのFDA承認化合物を用いてスクリニーング実験を行い、研究から僅か3ヶ月以内にCOVID19
の治療薬候補を見出しました。本研究成果はBioRxivにて発表されました。doi: 10.1101/2020.04.14.039925。

お気に入りの分子或いは調達サービスにより、分子ライブラリーをカスタマイズします。
お客様自身のニーズを満たすために、弊社の製品を数量、状態（乾燥状態/固体或いはDMSO）等で選択できます。

FDA-approved & Passed Phase I Drug Library内容

Download theFDA-approved & Passed Phase I Drug Library - SDF
Download theFDA-approved & Passed Phase I Drug Library - XLSX
Download the Compound Library Usage Instructions- PDF

Selleckの分子ライブラリーが使用されている文献(73)

Selleck化合物ライブラリー使用例

  • 肝癌研究におけるGPCR Compound Libraryの使用例

    Nature.2019;574(7777):268-272

  • 大腸癌研究におけるKinase Inhibitor Library の使用例

    Nat Commun. 2019 16;10(1):2197

  • 抗ウイルス研究におけるFDA-approved Drug Libraryの使用例

    Cell Res. 2019;29(9):739-753

  • 代謝研究におけるFDA-approved Drug Library使用例

    Mov Disord. 2019;34(3):323-334

  • 白血病研究におけるEpigenetics Compound Libraryの使用例

    Blood. 2019 17;134(16):1323-1336

  • 癌免疫研究におけるInhibitor Libraryの使用例

    Cancer Immunol Res.2017;5(9):790-803

製品特性＆メリット

・世界中で販売されている薬剤と、第1相臨床試験を通過した2880 種類の薬剤ライブラリー。HTS（High Throughput Screening） およびHCS（High Content Screening）に使用できます。

・既存の薬剤を用いて新たな適応症への効果を模索します。新薬開発よりも低コストで迅速な臨床効果が期待できます。

・第1相臨床試験で安全性が確認されました。

・腫瘍、心臓病、抗炎症、免疫、神経精神病、鎮痛などに関連しています。

・構造的に多様で、薬効および細胞透過性が確認されています。

・構造、IC50、お客様からのレビューなど豊富な情報があります

・NMRとHPLC検査で製品の高純度を保証しています。

製品詳細情報

調合： 2550 compounds pre-dissolved in 10mM DMSO, 229 compounds pre-dissolved in 10mM water, 84 compounds pre-dissolved in 2mM DMSO and 17 compounds pre-dissolved in 2mM water
ケース： 96/384 Well Format Sample Storage Tube With Screw Cap and Optional 2D Barcode
安定性： in DMSO
in DMSO
出荷方式： ブルーアイス物流
包装： 不活性ガス（Inert gas）

FDA-approved & Passed Phase I Drug Library组成

HTS パートナ

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