Immunology & Inflammation related

  • 阻害剤の選択性比較
  • 溶解度
カタログ番号 製品カタログ 溶解度(25°C)
DMSO アルコール
S2286 Cyclosporin A <1 mg/mL 100 mg/mL 100 mg/mL
S5004 Pimecrolimus <1 mg/mL 100 mg/mL 100 mg/mL
S1211 Imiquimod <1 mg/mL 1 mg/mL <1 mg/mL
S3032 Bindarit <1 mg/mL 64 mg/mL 64 mg/mL
S1407 Bimatoprost <1 mg/mL 36 mg/mL 83 mg/mL
S3622 Diammonium Glycyrrhizinate 100 mg/mL 100 mg/mL <1 mg/mL
S3608 Demethylzeylasteral (T-96) <1 mg/mL 96 mg/mL 33 mg/mL
S4753 Ganoderic acid A <1 mg/mL 100 mg/mL 100 mg/mL
S8522 Compstatin 100 mg/mL -1 mg/mL -1 mg/mL
S8141 Cl-amidine 70 mg/mL 84 mg/mL 84 mg/mL
S8291 Atractylenolide I <1 mg/mL 46 mg/mL 46 mg/mL
S8301 AS101 <1 mg/mL 62 mg/mL <1 mg/mL
S1439 Tranilast <1 mg/mL 66 mg/mL <1 mg/mL
S1737 Prednisolone <1 mg/mL 72 mg/mL 10 mg/mL
S1622 Prednisone <1 mg/mL 71 mg/mL <1 mg/mL
S4169 Teriflunomide <1 mg/mL 32 mg/mL ,1 mg/mL
S2413 Geniposidic acid <1 mg/mL 16 mg/mL 2 mg/mL
S1508 Alprostadil <1 mg/mL 71 mg/mL 71 mg/mL
S1733 Methylprednisolone <1 mg/mL 75 mg/mL 2 mg/mL
S1939 (-)-Tetramisole 48 mg/mL <1 mg/mL <1 mg/mL
S2787 Laquinimod <1 mg/mL 61 mg/mL 1 mg/mL
S1681 Mesalamine <1 mg/mL 31 mg/mL 31 mg/mL
S2910 Tempol 34 mg/mL 34 mg/mL 34 mg/mL
S1679 Flurbiprofen <1 mg/mL 49 mg/mL 49 mg/mL
S1829 Pranlukast <1 mg/mL 11 mg/mL <1 mg/mL
S1514 Cyclosporine <1 mg/mL 100 mg/mL 100 mg/mL
S1576 Sulfasalazine <1 mg/mL 80 mg/mL <1 mg/mL
S1654 Phenylbutazone <1 mg/mL 62 mg/mL 62 mg/mL
S2512 Tenoxicam <1 mg/mL 68 mg/mL <1 mg/mL
S3062 Diclofenac Potassium 10 mg/mL 69 mg/mL <1 mg/mL
S7515 VGX-1027 <1 mg/mL 41 mg/mL 41 mg/mL
S4098 Halcinonide <1 mg/mL 90 mg/mL 4 mg/mL
S1823 Fenoprofen Calcium <1 mg/mL 105 mg/mL 10 mg/mL
S4268 Flufenamic acid <1 mg/mL 56 mg/mL 56 mg/mL
S4529 Idramantone 33 mg/mL 33 mg/mL 33 mg/mL
S7211 PF-04418948 <1 mg/mL 81 mg/mL <1 mg/mL
S4152 Ethamsylate 53 mg/mL 53 mg/mL <1 mg/mL
S4165 Benzydamine HCl 69 mg/mL 69 mg/mL 69 mg/mL
S4170 Coumarin <1 mg/mL 29 mg/mL 29 mg/mL
S7809 85 mg/mL <1 mg/mL 40 mg/mL
S2400 Rheic Acid <1 mg/mL <1 mg/mL <1 mg/mL
S4188 Sasapyrine <1 mg/mL 52 mg/mL 52 mg/mL
S7448 CORM-3 <1 mg/mL 38 mg/mL <1 mg/mL
S4682 Loxoprofen <1 mg/mL 49 mg/mL 49 mg/mL
S7516 Y-320 <1 mg/mL 11 mg/mL <1 mg/mL
S3027 Fenoprofen calcium hydrate <1 mg/mL 48 mg/mL 18 mg/mL
S8097 C-DIM12 <1 mg/mL 71 mg/mL 71 mg/mL
S2350 Rutin <1 mg/mL 100 mg/mL 2 mg/mL
S7434 TAPI-1 60 mg/mL 99 mg/mL 99 mg/mL
S4690 Escin <1 mg/mL 66 mg/mL <1 mg/mL
製品コード 製品説明 文献中の使用例 お客様のフィードバック
S2286

Cyclosporin A

Cyclosporin A is an antilymphocytic agent, competitively binds to and inhibits calcineurin.

S5004

Pimecrolimus

Pimecrolimus, like all ascomycins, is an immunophilin ligand, which binds specifically to the cytosolic receptor, immunophilin macrophilin-12.

S1211

Imiquimod

Imiquimod is a novel synthetic agent with immune response modifying activity.

S3032

Bindarit

ビンダリットは、独特な抗炎症性活動が単球走化性タンパク質MCP-1/CCL2、MCP-3/CCL7とMCP-2/CCL8を含む炎症性ケモカインの亜族の選択的な抑制のためにある最初の合成物です。

S1407

Bimatoprost

Bimatoprost is a prostaglandin analog used topically (as eye drops) to control the progression of glaucoma and in the management of ocular hypertension.

A2009

Rituximab

S3622

Diammonium Glycyrrhizinate

S3608

Demethylzeylasteral (T-96)

S8559

INF39

A2001

Ipilimumab

Ipilimumab is an immunomodulatory monoclonal antibody directed against the cell surface antigen CTLA-4 and also a type of immune checkpoint inhibitor.

S4753

Ganoderic acid A

S8522

Compstatin

S8141

Cl-amidine

S8291

Atractylenolide I

S8301

AS101

S1439

Tranilast

Tranilast is an antiallergic compound.

S1737

Prednisolone

Prednisolone(Hydroretrocortine) is a synthetic glucocorticoid with anti-inflammatory and immunomodulating properties.

S1622

Prednisone

Prednisone (Adasone) is a synthetic corticosteroid agent that is particularly effective as an immunosuppressant compound.

S4169

Teriflunomide

Teriflunomideは、免疫調節剤として用いられる酵素ジヒドロデヒドロゲナーゼを遮断することによってレフルノミド、阻害ピリミジンデノボ合成の活性代謝産物です。

S2413

Geniposidic acid

Geniposidic acid is an effective anticancer and radioprotection agent.

S1508

Alprostadil

Alprostadil is used as a drug in the treatment of erectile dysfunction and has vasodilatory properties.

S1733

Methylprednisolone

Methylprednisolone is a synthetic glucocorticoid receptor agonist, used to achieve prompt suppression of inflammation.

S1939

(-)-Tetramisole

Levamisole Hydrochloride(Ergamisol)is an antihelminthic drug that has been tried experimentally in rheumatic disorders where it apparently restores the immune response by increasing macrophage chemotaxis and T-lymphocyte function.

S2787

Laquinimod

Laquinimod (ABR-215062) は、強力な免疫調節物質です。

S1681

Mesalamine

Mesalamine is an anti-inflammatory compound.

S2910

Tempol

TEMPOL is a superoxide scavenger that displays neuroprotective, anti-inflammatory and analgesic effects.

S1679

Flurbiprofen

Flurbiprofen is a member of the phenylalkanoic acid derivative family of non-steroidal anti-inflammatory drugs (NSAIDs).

S1829

Pranlukast

Pranlukast is an orally administered, and selective antagonist of the cysteinyl leukotrienes (LT) C(4), LTD(4) and LTE(4), used in the prophylactic treatment of chronic bronchial asthma.

S1514

Cyclosporine

Cyclosporine (Neoral) is an immunosuppressant drug.

S1576

Sulfasalazine

Sulfasalazine is a sulfa agent and a derivative of mesalazine used primarily as an anti-inflammatory agent.

S1654

Phenylbutazone

Phenylbutazone(Butazolidin, Butatron) is used as a non-steroidal anti-inflammatory agent for the treatment of chronic pain, including the symptoms of arthritis.

S2512

Tenoxicam

Tenoxicam is a good HO. radicals scavenger with an IC50 of 56.7 μM

S3062

Diclofenac Potassium

Diclofenac potassium is a nonsteroidal anti-inflammatory drug taken to reduce inflammation and as an analgesic reducing pain in certain conditions.

S7515

VGX-1027

VGX-1027 is an orally active immunomodulator. Phase1.

S4098

Halcinonide

Halcinonide is a high potency corticosteroid used in topical preparations as an anti-inflammatory agent.

S1823

Fenoprofen Calcium

Fenoprofen calcium is a nonsteroidal, anti-inflammatory antiarthritic agent.

S4268

Flufenamic acid

Flufenamic Acid is an anti-inflammatory agent, and also acts as an ion channel modulator.

S4529

Idramantone

S7211

PF-04418948

PF-04418948 is a potent and selective prostaglandin EP₂ receptor antagonist with IC50 of 16 nM. Phase 1.

S4152

Ethamsylate

Ethamsylateは生とプロスタグランジンの作用を阻害する止血薬であり、毛細血管内皮抵抗などと血小板の接着性を向上させます。

S4165

Benzydamine HCl

Benzydamine hydrochlorideは、抗炎症、鎮痛、解熱及び局所麻酔薬活性を有する局所用非ステロイド系抗炎症薬(NSAID)です。

S4170

Coumarin

Coumarinは肝毒性と発がん性を有する二次植物化学物質です。

S7809

S2400

Rheic Acid

Rhein(Monorhein; NSC 38629; Rheic acid; Rheinic acid) is a constituent of rhubarb which was isolated from the fresh rhizome of Rheum coreanum Nakai.

S4188

Sasapyrine

Sasapyrine (salsalate)は非ステロイド経口抗炎症剤です。

S7448

CORM-3

CORM-3 is a water-soluble carbon monoxide-releasing molecule with anti-inflammatory and cardioprotective activity.

S4682

Loxoprofen

Loxoprofenはプロピオン酸派生物に於いて、1種の非ステロイド性の(non-steroidal)消炎薬です。

S7516

Y-320

Y-320 is an orally active immunomodulator, and inhibits IL-17 production by CD4 T cells stimulated with IL-15 with IC50 of 20 to 60 nM.

S3027

Fenoprofen calcium hydrate

フェノプロフェン・カルシウム水和物(Nalfon)は、非ステロイド性の抗炎症剤(NSAID)です。

S4706

Eugenol

S8097

C-DIM12

S4709

Latanoprost

S2350

Rutin

Rutin, a flavonol glycoside found in many plants, including buckwheat; tobacco; forsythia; hydrangea; viola, etc.

S7434

TAPI-1

TAPI-1 is an ADAM17/TACE inhibitor, which blocks shedding of cytokine receptors.

S4690

Escin

S4524

2-Ethoxybenzamide