ACE
阻害剤の選択性比較
| カタログ番号 | 製品カタログ | 溶解度(25°C) | ||
|---|---|---|---|---|
| 水 | DMSO | アルコール | ||
| S1793 | Ramipril | <1 mg/mL | 83 mg/mL | '83 mg/mL |
| S1941 | Enalapril Maleate | <1 mg/mL | 99 mg/mL | ''4 mg/mL |
| S2051 | Captopril | 2 mg/mL | 43 mg/mL | '43 mg/mL |
| S2076 | Lisinopril dihydrate | 20 mg/mL | <1 mg/mL | ''''<1 mg/mL |
| S2079 | Moexipril HCl | <1 mg/mL | 20 mg/mL | ''<1 mg/mL |
| S2099 | Temocapril HCl | <1 mg/mL | 103 mg/mL | '103 mg/mL |
| S2100 | Temocapril | <1 mg/mL | 95 mg/mL | ''95 mg/mL |
| S2109 | Imidapril HCl | 54 mg/mL | 88 mg/mL | '29 mg/mL |
| S5728 | Delapril Hydrochloride | <1 mg/mL | 98 mg/mL | ''25 mg/mL |
| S6468 | Trandolapril | <1 mg/mL | 86 mg/mL | '43 mg/mL |
| S2095 | Fosinopril Sodium | 117 mg/mL | <1 mg/mL | ''4 mg/mL |
| S1733 | Methylprednisolone | <1 mg/mL | 75 mg/mL | '''''2 mg/mL |
| S4104 | Diminazene Aceturate | 100 mg/mL | 19 mg/mL | <1 mg/mL |
ACE製品
| 製品コード | 製品説明 | 文献中Selleckの製品使用例 | お客様のフィードバック |
|---|---|---|---|
| S1793 |
RamiprilRamipril is an angiotensin-converting enzyme (ACE) inhibitor with IC50 of 5 nM. |
||
| S1941 |
Enalapril MaleateEnalapril (MK-421) Maleate is an angiotensin-converting enzyme (ACE) inhibitor, used in the treatment of hypertension, diabetic nephropathy, and chronic heart failure. |
||
| S2051 |
CaptoprilCaptopril is an angiotensin-converting enzyme (ACE) inhibitor with IC50 of 6 nM. |
||
| S2076 |
Lisinopril dihydrateLisinopril dihydrate is an angiotensin-converting enzyme (ACE) inhibitor, used in treatment of hypertension, congestive heart failure, and heart attacks, and also in preventing renal and retinal complications of diabetes. |
||
| S2079 |
Moexipril HClMoexipril HCl is a potent orally active nonsulfhydryl angiotensin converting enzyme (ACE) inhibitor, used for the treatment of hypertension and congestive heart failure. |
||
| S2099 |
Temocapril HClTemocapril HCl is the hydrochloride of Temocapril, which is a long-acting angiotensin-converting enzyme (ACE) inhibitor, used for the treatment of hypertension. |
||
| S2100 |
TemocaprilTemocapril (CS-622) is a long-acting angiotensin-converting enzyme (ACE) inhibitor, used for the treatment of hypertension. |
||
| S2109 |
Imidapril HClImidapril HCl is an angiotensin-converting enzyme (ACE) inhibitor with IC50 of 2.6 nM, used for the treatment of hypertension. |
||
| S5728 |
Delapril HydrochlorideDelapril Hydrochloride (Alindapril) is the hydrochloride salt form of delapril, which is a lipophilic, non-sulfhydryl angiotensin-converting enzyme (ACE) inhibitor with antihypertensive activity. |
||
| S6468 |
TrandolaprilTrandolapril is a newly developed angiotensin-converting enzyme (ACE) inhibitor that is rapidly hydrolyzed mainly in the liver to its biologically active metabolite trandolaprilat. |
||
| S2095 |
Fosinopril SodiumFosinopril Sodium (SQ28555) is the ester prodrug of an angiotensin-converting enzyme (ACE) inhibitor, used for the treatment of hypertension and some types of chronic heart failure. |
||
| S1733 |
MethylprednisoloneMethylprednisolone (NSC-19987) is a synthetic glucocorticoid receptor agonist, used to achieve prompt suppression of inflammation. Methylprednisolone activates ACE2 and reduces IL-6 levels, thus improves severe or critical COVID-19. Methylprednisolone markedly reduces autophagy and apoptosis. |
Motor disturbances of the rat hindlimbs after SCI, using an inclined plane test. Key: ◇ = PBS group; ■ = Sal B group; ▲ = methylprednisolone group.
|
|
| S4104 |
Diminazene AceturateDiminazene is a di-amidine also known as 4,4-(1-Triazene–1,3–diyl)bis(benzenecarboximidamide), used as an effective trypanocidal agent. |
| 製品コード | 製品説明 | 文献中Selleckの製品使用例 | お客様のフィードバック |
|---|---|---|---|
| S1793 |
RamiprilRamipril is an angiotensin-converting enzyme (ACE) inhibitor with IC50 of 5 nM. |
||
| S1941 |
Enalapril MaleateEnalapril (MK-421) Maleate is an angiotensin-converting enzyme (ACE) inhibitor, used in the treatment of hypertension, diabetic nephropathy, and chronic heart failure. |
||
| S2051 |
CaptoprilCaptopril is an angiotensin-converting enzyme (ACE) inhibitor with IC50 of 6 nM. |
||
| S2076 |
Lisinopril dihydrateLisinopril dihydrate is an angiotensin-converting enzyme (ACE) inhibitor, used in treatment of hypertension, congestive heart failure, and heart attacks, and also in preventing renal and retinal complications of diabetes. |
||
| S2079 |
Moexipril HClMoexipril HCl is a potent orally active nonsulfhydryl angiotensin converting enzyme (ACE) inhibitor, used for the treatment of hypertension and congestive heart failure. |
||
| S2099 |
Temocapril HClTemocapril HCl is the hydrochloride of Temocapril, which is a long-acting angiotensin-converting enzyme (ACE) inhibitor, used for the treatment of hypertension. |
||
| S2100 |
TemocaprilTemocapril (CS-622) is a long-acting angiotensin-converting enzyme (ACE) inhibitor, used for the treatment of hypertension. |
||
| S2109 |
Imidapril HClImidapril HCl is an angiotensin-converting enzyme (ACE) inhibitor with IC50 of 2.6 nM, used for the treatment of hypertension. |
||
| S5728 |
Delapril HydrochlorideDelapril Hydrochloride (Alindapril) is the hydrochloride salt form of delapril, which is a lipophilic, non-sulfhydryl angiotensin-converting enzyme (ACE) inhibitor with antihypertensive activity. |
||
| S6468 |
TrandolaprilTrandolapril is a newly developed angiotensin-converting enzyme (ACE) inhibitor that is rapidly hydrolyzed mainly in the liver to its biologically active metabolite trandolaprilat. |
||
| S2095 |
Fosinopril SodiumFosinopril Sodium (SQ28555) is the ester prodrug of an angiotensin-converting enzyme (ACE) inhibitor, used for the treatment of hypertension and some types of chronic heart failure. |
| 製品コード | 製品説明 | 文献中Selleckの製品使用例 | お客様のフィードバック |
|---|---|---|---|
| S1733 |
MethylprednisoloneMethylprednisolone (NSC-19987) is a synthetic glucocorticoid receptor agonist, used to achieve prompt suppression of inflammation. Methylprednisolone activates ACE2 and reduces IL-6 levels, thus improves severe or critical COVID-19. Methylprednisolone markedly reduces autophagy and apoptosis. |
2020, 10.1002/dta.2917 2017, 23(4):424-428 2014, 13 (1): 53-59 |
Motor disturbances of the rat hindlimbs after SCI, using an inclined plane test. Key: ◇ = PBS group; ■ = Sal B group; ▲ = methylprednisolone group.
|
| S4104 |
Diminazene AceturateDiminazene is a di-amidine also known as 4,4-(1-Triazene–1,3–diyl)bis(benzenecarboximidamide), used as an effective trypanocidal agent. |
2020, 10.1152/ajplung.00025.2020 |
