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NPY receptor

亜型選択性的な製品

NPY receptor製品

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  • NPY receptor拮抗剤(4)
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製品コード 製品名称 製品説明 文献中Selleckの製品使用例 お客様のフィードバック
E0014 BIBO 3304 Trifluoroacetate BIBO 3304 Trifluoroacetate (BIBO-3304 TFA) is a novel neuropeptide Y Y1 receptor (NPY1R) antagonist with IC50 values of 0.38 nM and 0.72 nM for human Y1 receptor and rat Y1 receptor, respectively. BIBO 3304 shows low affinity for the human Y2 receptor, human and rat Y4 receptor as well as for the human and rat Y5 receptor (IC50 values >1000 nM).
Adv Sci (Weinh), 2021, e2100808
E2134 WAY-639889 WAY-639889 is a bioactive compound relative to neuropeptide Y-5.
S0124 CGP71683 hydrochloride CGP71683 hydrochloride (CGP71683A) is a competitive and sellective neuropeptide Y receptor type 5 (Y5 receptor) antagonist with Ki of 1.3 nM.
S6416 JNJ 31020028 JNJ 31020028 is a novel neuropeptide Y Y2 receptor antagonist which bound with high affinity with human and rat Y2 receptor (pIC50=8.07±0.05 for human Y2 receptor, and pIC50=8.22±0.06 for rat Y2 receptor) and >100-fold selective versus human Y1, Y4, and Y5 receptors.
E0014 BIBO 3304 Trifluoroacetate BIBO 3304 Trifluoroacetate (BIBO-3304 TFA) is a novel neuropeptide Y Y1 receptor (NPY1R) antagonist with IC50 values of 0.38 nM and 0.72 nM for human Y1 receptor and rat Y1 receptor, respectively. BIBO 3304 shows low affinity for the human Y2 receptor, human and rat Y4 receptor as well as for the human and rat Y5 receptor (IC50 values >1000 nM).
Adv Sci (Weinh), 2021, e2100808
E2134 WAY-639889 WAY-639889 is a bioactive compound relative to neuropeptide Y-5.
S0124 CGP71683 hydrochloride CGP71683 hydrochloride (CGP71683A) is a competitive and sellective neuropeptide Y receptor type 5 (Y5 receptor) antagonist with Ki of 1.3 nM.
S6416 JNJ 31020028 JNJ 31020028 is a novel neuropeptide Y Y2 receptor antagonist which bound with high affinity with human and rat Y2 receptor (pIC50=8.07±0.05 for human Y2 receptor, and pIC50=8.22±0.06 for rat Y2 receptor) and >100-fold selective versus human Y1, Y4, and Y5 receptors.

NPY receptor阻害剤の選択性比較

Tags: NPY receptor inhibitor|NPY receptor agonist|NPY receptor activator|NPY receptor inducer|NPY receptor antagonist|NPY receptor signaling pathway|NPY receptor assay kit