SUMO

阻害剤の選択性比較

カタログ番号 製品カタログ 溶解度(25°C)
DMSO アルコール
S4922 NSC 632839 <1 mg/mL 7 mg/mL ''''<1 mg/mL
S8829 Subasumstat (TAK-981) <1 mg/mL 100 mg/mL ''<1 mg/mL
S8696 2-D08 <1 mg/mL 54 mg/mL '<1 mg/mL
S9432 Ginkgolic Acid -1 mg/mL 69 mg/mL -1 mg/mL
S9445 Ginkgolic Acid (C13:0) -1 mg/mL 64 mg/mL -1 mg/mL
S9159 momordin-Ic -1 mg/mL 100 mg/mL -1 mg/mL

亜型選択性的な製品

SUMO製品

製品コード 製品説明 文献中Selleckの製品使用例 お客様のフィードバック
S4922

NSC 632839

NSC 632839 is not only a DUB inhibitor, but also a deSUMOylase inhibitor, it inhibits USP2, USP7, and SENP2 with EC50 of 45 μM, 37 μM, and 9.8 μM, respectively.

S8829

Subasumstat (TAK-981)

Subasumstat (TAK-981) is a novel, selective inhibitor of the SUMOylation enzymatic cascade with potential immune-activating and antineoplastic activities.

S8696

2-D08

2-D08 (2',3',4'-trihydroxy flavone) is a cell permeable, mechanistically unique inhibitor of protein sumoylation.

S9432

Ginkgolic Acid

Ginkgolic acid, toxic phenolic compounds present in the fruits and leaves of Ginkgo biloba L., is a potent sumoylation inhibitor also reported to inhibit histone acetylation transferase (HAT).

S9445

Ginkgolic Acid (C13:0)

Ginkgolic Acid (C13:0) is a natural anticariogenic agent in Ginkgo biloba L. that exhibits antimicrobial activity against S. mutans and suppresses the specific virulence factors associated with its cariogenicity. Ginkgolic acid is a potent sumoylation inhibitor and reported to inhibit histone acetylation transferase (HAT).

S9159

momordin-Ic

Momordin Ic, a natural triterpenoid saponin, is a novel SENP1 (SUMO-specific protease 1) inhibitor that inhibited proliferation of prostate cancer cells in vitro and in vivo.

製品コード 製品説明 文献中Selleckの製品使用例 お客様のフィードバック
S4922

NSC 632839

NSC 632839 is not only a DUB inhibitor, but also a deSUMOylase inhibitor, it inhibits USP2, USP7, and SENP2 with EC50 of 45 μM, 37 μM, and 9.8 μM, respectively.

S8829

Subasumstat (TAK-981)

Subasumstat (TAK-981) is a novel, selective inhibitor of the SUMOylation enzymatic cascade with potential immune-activating and antineoplastic activities.

S8696

2-D08

2-D08 (2',3',4'-trihydroxy flavone) is a cell permeable, mechanistically unique inhibitor of protein sumoylation.

S9432

Ginkgolic Acid

Ginkgolic acid, toxic phenolic compounds present in the fruits and leaves of Ginkgo biloba L., is a potent sumoylation inhibitor also reported to inhibit histone acetylation transferase (HAT).

S9445

Ginkgolic Acid (C13:0)

Ginkgolic Acid (C13:0) is a natural anticariogenic agent in Ginkgo biloba L. that exhibits antimicrobial activity against S. mutans and suppresses the specific virulence factors associated with its cariogenicity. Ginkgolic acid is a potent sumoylation inhibitor and reported to inhibit histone acetylation transferase (HAT).

S9159

momordin-Ic

Momordin Ic, a natural triterpenoid saponin, is a novel SENP1 (SUMO-specific protease 1) inhibitor that inhibited proliferation of prostate cancer cells in vitro and in vivo.

Tags: SUMO Inhibition | SUMO antibody | SUMO inhibitors | SUMO modulation