ADAM10

ADAM10製品

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  • ADAM10阻害剤 (1)
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製品コード 製品名称 製品説明 文献中Selleckの製品使用例 お客様のフィードバック
S8660 GI254023X GI254023X (GI 4023, SRI028594) is a selective inhibitor of ADAM10 with 100-fold selectivity for ADAM10 over ADAM17. The IC50 values for recombinant ADAM10 amd ADAM17 are 5.3 nM and 541 nM, respectively. GI254023X can inhibit MMP9.
Signal Transduct Target Ther, 2025, 10(1):387
Cell Death Dis, 2025, 16(1):34
Alzheimers Res Ther, 2024, 16(1):160
S8660 GI254023X GI254023X (GI 4023, SRI028594) is a selective inhibitor of ADAM10 with 100-fold selectivity for ADAM10 over ADAM17. The IC50 values for recombinant ADAM10 amd ADAM17 are 5.3 nM and 541 nM, respectively. GI254023X can inhibit MMP9.
Signal Transduct Target Ther, 2025, 10(1):387
Cell Death Dis, 2025, 16(1):34
Alzheimers Res Ther, 2024, 16(1):160