Parasite

阻害剤の選択性比較

カタログ番号 製品カタログ 溶解度(25°C)
DMSO アルコール
S2468 Fenbendazole <1 mg/mL 4 mg/mL '<1 mg/mL
S1837 Flubendazole <1 mg/mL 3 mg/mL '<1 mg/mL
S7379 E-64 11 mg/mL 71 mg/mL '<1 mg/mL
S4044 Toltrazuril <1 mg/mL 85 mg/mL '<1 mg/mL
S3741 Benznidazole <1 mg/mL 52 mg/mL ''5 mg/mL
S0081 DDD107498 succinate ' mg/mL
S4422 Nitenpyram 54 mg/mL 54 mg/mL '54 mg/mL
S3889 Arteether -1 mg/mL 62 mg/mL ''-1 mg/mL
S5557 Aklomide -1 mg/mL 40 mg/mL '-1 mg/mL
S4564 Diethylcarbamazine citrate 78 mg/mL 78 mg/mL ''30 mg/mL
S5247 Selamectin -1 mg/mL 100 mg/mL ''-1 mg/mL

Parasite製品

製品コード 製品説明 文献中Selleckの製品使用例 お客様のフィードバック
S2468

Fenbendazole

Fenbendazole is a broad spectrum benzimidazole anthelmintic used against gastrointestinal parasites with an IC50 of about 0.01 μg/mL.

S1837

Flubendazole

Flubendazole (Flumoxanal, NSC 313680) is an autophagy inducer by targeting Atg4B, used to treat internal parasite and worm infection.

S7379

E-64

E-64 is an irreversible and selective cysteine protease inhibitor, and also inhibits papain, calpain, and cathepsins B and H, but not serine proteases or aspartic proteases. The IC50 for papain is 9 nM. E-64 induces oxidative stress and apoptosis in Filarial Parasite.

S4044

Toltrazuril

Toltrazuril is an antiprotozoal agent that acts upon Coccidia parasites.

S3741

Benznidazole

Benznidazole (Radanil) is a nitroimidazole derivative having an antiprotozoal activity by interfering with parasite protein biosynthesis, influencing cytokines production and stimulating host phagocytosis.

S0081

DDD107498 succinate

DDD107498 succinate (DDD-498 succinate) is a potent and orally active antimalarial agent. DDD107498 succinate inhibits multiple life-cycle stages of the parasite with EC50 of 1 nM against P. falciparum 3D7. DDD107498 succinate inhibits protein synthesis by targeting eEF2/CaMKIII with EC50 of 2 nM for WT-PfeEF2.

S4422

Nitenpyram

Nitenpyram is a nicotinic acetylcholine receptor (AchR) agonist, used as veterinary medicine to treat parasites of livestock and pets.

S3889

Arteether

Arteether is a well-known antimalarial drug which acts by producing free radicals within the malarial parasite.

S5557

Aklomide

Aklomide (2-Chloro-4-nitrobenzamide) is a coccidiostat and used to fight disease, parasites and insects that infest poultry.

S4564

Diethylcarbamazine citrate

Diethylcarbamazine citrate is an inhibitor of arachidonic acid metabolism in filarial microfilaria and is highly specific for several parasites and does not contain any toxic metallic elements.

S5247

Selamectin

Selamectin (UK-124114) is a novel macrocyclic lactone of the avermectin class. It paralyses and/or kills a wide range of invertebrate parasites through interference with their chloride channel conductance causing disruption of normal neurotransmission and has adulticidal, ovicidal and larvicidal activity against fleas.

製品コード 製品説明 文献中Selleckの製品使用例 お客様のフィードバック
S2468

Fenbendazole

Fenbendazole is a broad spectrum benzimidazole anthelmintic used against gastrointestinal parasites with an IC50 of about 0.01 μg/mL.

S1837

Flubendazole

Flubendazole (Flumoxanal, NSC 313680) is an autophagy inducer by targeting Atg4B, used to treat internal parasite and worm infection.

S7379

E-64

E-64 is an irreversible and selective cysteine protease inhibitor, and also inhibits papain, calpain, and cathepsins B and H, but not serine proteases or aspartic proteases. The IC50 for papain is 9 nM. E-64 induces oxidative stress and apoptosis in Filarial Parasite.

S4044

Toltrazuril

Toltrazuril is an antiprotozoal agent that acts upon Coccidia parasites.

S3741

Benznidazole

Benznidazole (Radanil) is a nitroimidazole derivative having an antiprotozoal activity by interfering with parasite protein biosynthesis, influencing cytokines production and stimulating host phagocytosis.

S0081

DDD107498 succinate

DDD107498 succinate (DDD-498 succinate) is a potent and orally active antimalarial agent. DDD107498 succinate inhibits multiple life-cycle stages of the parasite with EC50 of 1 nM against P. falciparum 3D7. DDD107498 succinate inhibits protein synthesis by targeting eEF2/CaMKIII with EC50 of 2 nM for WT-PfeEF2.

S4422

Nitenpyram

Nitenpyram is a nicotinic acetylcholine receptor (AchR) agonist, used as veterinary medicine to treat parasites of livestock and pets.

S3889

Arteether

Arteether is a well-known antimalarial drug which acts by producing free radicals within the malarial parasite.

S5557

Aklomide

Aklomide (2-Chloro-4-nitrobenzamide) is a coccidiostat and used to fight disease, parasites and insects that infest poultry.

S4564

Diethylcarbamazine citrate

Diethylcarbamazine citrate is an inhibitor of arachidonic acid metabolism in filarial microfilaria and is highly specific for several parasites and does not contain any toxic metallic elements.

S5247

Selamectin

Selamectin (UK-124114) is a novel macrocyclic lactone of the avermectin class. It paralyses and/or kills a wide range of invertebrate parasites through interference with their chloride channel conductance causing disruption of normal neurotransmission and has adulticidal, ovicidal and larvicidal activity against fleas.