Serine Protease

阻害剤の選択性比較

カタログ番号 製品カタログ 溶解度(25°C)
DMSO アルコール
S1386 Nafamostat Mesylate 53 mg/mL 20 mg/mL <1 mg/mL
S3025 PMSF <1 mg/mL 35 mg/mL 15 mg/mL
S2101 Gabexate Mesylate 12 mg/mL 83 mg/mL 83 mg/mL
S7218 Alvelestat (AZD9668) <1 mg/mL 100 mg/mL <1 mg/mL
S7378 AEBSF HCl 20 mg/mL 47 mg/mL 47 mg/mL
S7380 Leupeptin Hemisulfate 95 mg/mL 95 mg/mL 95 mg/mL
S8457 UK-371804 HCl <1 mg/mL 30 mg/mL <1 mg/mL
S4666 Sivelestat sodium tetrahydrate <1 mg/mL 100 mg/mL 100 mg/mL
S8136 Sivelestat (ONO-5046) <1 mg/mL 86 mg/mL 86 mg/mL
S7377 Aprotinin 100 mg/mL -1 mg/mL -1 mg/mL

Serine Protease製品

製品コード 製品説明 文献中Selleckの製品使用例 お客様のフィードバック
S1386

Nafamostat Mesylate

Nafamostat mesilate is a synthetic serine protease inhibitor, used as an anticoagulant during hemodialysis.

S3025

PMSF

PMSF is an irreversible serine/cysteine protease inhibitor.

S2101

Gabexate Mesylate

Gabexate Mesylate is a serine protease inhibitor with IC50 of 0.19 μM which is used therapeutically in the treatment of pancreatitis and disseminated intravascular coagulation.

S7218

Alvelestat (AZD9668)

Alvelestat (AZD9668) is an oral, highly selective inhibitor of neutrophil elastase (NE) with IC50 and Ki of 12 nM and 9.4 nM, at least 600-fold more selective over other serine proteases. Phase 2.

S7378

AEBSF HCl

AEBSF HCl is a broad spectrum, irreversible serine protease inhibitor.

S7380

Leupeptin Hemisulfate

Leupeptin Hemisulfate is a reversible inhibitor of serine and cysteine proteases. It inhibits cathepsin B (Ki = 6 nM), calpain (Ki = 10 nM), trypsin (Ki = 35 nM), plasmin (Ki = 3.4 μM), and kallikrein (Ki = 19 μM), and has no effect against chymotrypsin, elastase, renin, or pepsin.

S8457

UK-371804 HCl

UK-371804 is a potent and selective urokinase-type plasmogen activator (uPA) inhibitor with excellent enzyme potency (Ki=10 nM) and selectivity profile (4000-fold versus tPA and 2700-fold versus plasmin).

S4666

Sivelestat sodium tetrahydrate

Sivelestat sodium tetrahydrate is a competitive inhibitor of human neutrophil elastase, also inhibits leukocyte elastase obtained from rabbit, rat, hamster and mouse.

S8136

Sivelestat (ONO-5046)

Sivelestat is a potent and selective inhibitor of neutrophil elastase with IC50 of 44nM. It almost shows no activity at a range of other proteases.

S7377

Aprotinin

Aprotinin is a small protein serine protease inhibitor, used to reduce perioperative blood loss and transfusion.

製品コード 製品説明 文献中Selleckの製品使用例 お客様のフィードバック
S1386

Nafamostat Mesylate

Nafamostat mesilate is a synthetic serine protease inhibitor, used as an anticoagulant during hemodialysis.

S3025

PMSF

PMSF is an irreversible serine/cysteine protease inhibitor.

S2101

Gabexate Mesylate

Gabexate Mesylate is a serine protease inhibitor with IC50 of 0.19 μM which is used therapeutically in the treatment of pancreatitis and disseminated intravascular coagulation.

S7218

Alvelestat (AZD9668)

Alvelestat (AZD9668) is an oral, highly selective inhibitor of neutrophil elastase (NE) with IC50 and Ki of 12 nM and 9.4 nM, at least 600-fold more selective over other serine proteases. Phase 2.

S7378

AEBSF HCl

AEBSF HCl is a broad spectrum, irreversible serine protease inhibitor.

S7380

Leupeptin Hemisulfate

Leupeptin Hemisulfate is a reversible inhibitor of serine and cysteine proteases. It inhibits cathepsin B (Ki = 6 nM), calpain (Ki = 10 nM), trypsin (Ki = 35 nM), plasmin (Ki = 3.4 μM), and kallikrein (Ki = 19 μM), and has no effect against chymotrypsin, elastase, renin, or pepsin.

S8457

UK-371804 HCl

UK-371804 is a potent and selective urokinase-type plasmogen activator (uPA) inhibitor with excellent enzyme potency (Ki=10 nM) and selectivity profile (4000-fold versus tPA and 2700-fold versus plasmin).

S4666

Sivelestat sodium tetrahydrate

Sivelestat sodium tetrahydrate is a competitive inhibitor of human neutrophil elastase, also inhibits leukocyte elastase obtained from rabbit, rat, hamster and mouse.

S8136

Sivelestat (ONO-5046)

Sivelestat is a potent and selective inhibitor of neutrophil elastase with IC50 of 44nM. It almost shows no activity at a range of other proteases.

S7377

Aprotinin

Aprotinin is a small protein serine protease inhibitor, used to reduce perioperative blood loss and transfusion.

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