κ-opioid receptor Selective 作動薬

製品コード 製品名 製品説明 Selective / Pan IC50 / Ki
S2322 (+)-Matrine Matrine((+)-Matrine) is an alkaloid found in plants from the Sophora family, which has a variety of pharmacological effects, including anti-cancer effects, and action as a kappa opioid receptor agonist. Selective
S1139 ADL5859 HCl ADL5859 HCl is a δ-opioid receptor agonist with Ki of 0.8 nM, selectivity against opioid receptor κ, μ, and weak inhibitory activity at the hERG channel. Phase 2. Pan κ-opioid receptor, Ki: 37 nM
Tags: κ-opioid receptor inhibitor | κ-opioid receptor activity | κ-opioid receptor phosphorylation | κ-opioid receptor mutation