GHSR
阻害剤の選択性比較
| カタログ番号 | 製品カタログ | 溶解度(25°C) | ||
|---|---|---|---|---|
| 水 | DMSO | アルコール | ||
| S6948 | Lanreotide | 100 mg/mL | 100 mg/mL | 100 mg/mL |
| S4980 | Anamorelin | <1 mg/mL | 100 mg/mL | 79 mg/mL |
| S1151 | Ibutamoren mesylate | 100 mg/mL | 100 mg/mL | 100 mg/mL |
| S0169 | Capromorelin tartrate | 100 mg/mL | 100 mg/mL | '''100 mg/mL |
GHSR製品
| 製品コード | 製品説明 | 文献中Selleckの製品使用例 | お客様のフィードバック |
|---|---|---|---|
| S6948新 |
LanreotideLanreotide (Laromustine, Angiopeptin, BIM 23014, Dermopeptin, Ipstyl, ITM-014, Somatulina, Somatuline, Lanreotidum), an analog of the native somatostatin peptide, is a physiological inhibitor of growth hormone (GH). Lanreotide also has antitumoral effects. |
||
| S4980 |
AnamorelinAnamorelin (ONO-7643, RC-1291, ST-1291) is an orally active, high-affinity, selective agonist of the ghrelin receptor with an EC50 value of 0.74 nM in the HEK293/GRLN FLIPR assay. |
||
| S1151 |
Ibutamoren mesylateA potent, orally active growth hormone (GH) secretagogue. |
||
| S0169 |
Capromorelin tartrateCapromorelin Tartrate (CP 424391-18), a member of the growth hormone secretagogue (GHS) class of drugs, is a ghrelin receptor agonist and a novel therapy for stimulation of appetite in dogs with Ki of 7 nM for hGHS-R1a and EC50 of 3 nM for rat pituicyte. |
| 製品コード | 製品説明 | 文献中Selleckの製品使用例 | お客様のフィードバック |
|---|---|---|---|
| S6948新 |
LanreotideLanreotide (Laromustine, Angiopeptin, BIM 23014, Dermopeptin, Ipstyl, ITM-014, Somatulina, Somatuline, Lanreotidum), an analog of the native somatostatin peptide, is a physiological inhibitor of growth hormone (GH). Lanreotide also has antitumoral effects. |
| 製品コード | 製品説明 | 文献中Selleckの製品使用例 | お客様のフィードバック |
|---|---|---|---|
| S4980 |
AnamorelinAnamorelin (ONO-7643, RC-1291, ST-1291) is an orally active, high-affinity, selective agonist of the ghrelin receptor with an EC50 value of 0.74 nM in the HEK293/GRLN FLIPR assay. |
2020, 10.1002/dta.2917 |
|
| S1151 |
Ibutamoren mesylateA potent, orally active growth hormone (GH) secretagogue. |
2021, 10.1021/acs.analchem.1c01083 |
|
| S0169 |
Capromorelin tartrateCapromorelin Tartrate (CP 424391-18), a member of the growth hormone secretagogue (GHS) class of drugs, is a ghrelin receptor agonist and a novel therapy for stimulation of appetite in dogs with Ki of 7 nM for hGHS-R1a and EC50 of 3 nM for rat pituicyte. |
2020, 10.1002/dta.2917 |
