グルココルチコイド受容体
阻害剤の選択性比較
| カタログ番号 | 製品カタログ | 溶解度(25°C) | ||
|---|---|---|---|---|
| 水 | DMSO | アルコール | ||
| S1322 | Dexamethasone (MK-125) | <1 mg/mL | 79 mg/mL | '''6 mg/mL |
| E0177 | Hydrocortisone sodium succinate | 97 mg/mL | 97 mg/mL | 24 mg/mL |
| S2606 | Mifepristone (RU486) | <1 mg/mL | 85 mg/mL | ''''19 mg/mL |
| S6608 | AL082D06 | <1 mg/mL | 10 mg/mL | <1 mg/mL |
| S1696 | Hydrocortisone (NSC 10483) | <1 mg/mL | 73 mg/mL | ''23 mg/mL |
| S1737 | Prednisolone (NSC-9900) | <1 mg/mL | 72 mg/mL | '''10 mg/mL |
| S1622 | Prednisone (NSC-10023) | <1 mg/mL | 71 mg/mL | '<1 mg/mL |
| S5489 | Prednisone acetate | <1 mg/mL | 27 mg/mL | ''<1 mg/mL |
| S5956 | Dexamethasone phosphate disodium | 100 mg/mL | <1 mg/mL | ''<1 mg/mL |
| S5973 | Methylprednisolone Acetate | <1 mg/mL | 86 mg/mL | ''<1 mg/mL |
| S5184 | Dexamethasone palmitate | <1 mg/mL | 100 mg/mL | ''100 mg/mL |
| S1669 | Loteprednol etabonate | <1 mg/mL | 93 mg/mL | 4 mg/mL |
| S1987 | Mometasone furoate | <1 mg/mL | 6 mg/mL | <1 mg/mL |
| S1992 | Fluticasone propionate | <1 mg/mL | 100 mg/mL | 5 mg/mL |
| S1733 | Methylprednisolone (NSC-19987) | <1 mg/mL | 75 mg/mL | '2 mg/mL |
| S1286 | Budesonide | <1 mg/mL | 86 mg/mL | 19 mg/mL |
| S1628 | Triamcinolone Acetonide | <1 mg/mL | 87 mg/mL | 13 mg/mL |
| S1689 | Meprednisone | <1 mg/mL | 75 mg/mL | 4 mg/mL |
| S1888 | Deflazacort | <1 mg/mL | 88 mg/mL | 12 mg/mL |
| S2470 | Fluocinolone Acetonide | <1 mg/mL | 90 mg/mL | 12 mg/mL |
| S1688 | Betamethasone Dipropionate | <1 mg/mL | 100 mg/mL | 66 mg/mL |
| S1690 | Betamethasone Valerate | <1 mg/mL | 95 mg/mL | 58 mg/mL |
| S2570 | Prednisolone Acetate | <1 mg/mL | 81 mg/mL | <1 mg/mL |
| S1500 | Betamethasone | <1 mg/mL | 79 mg/mL | 10 mg/mL |
| S4088 | Flumethasone | <1 mg/mL | 82 mg/mL | 6 mg/mL |
| S1701 | Desonide | <1 mg/mL | 83 mg/mL | 30 mg/mL |
| S2608 | Fluocinonide | <1 mg/mL | 99 mg/mL | <1 mg/mL |
| S2584 | Clobetasol propionate | <1 mg/mL | 93 mg/mL | 20 mg/mL |
| S1933 | Triamcinolone | <1 mg/mL | 78 mg/mL | 1 mg/mL |
| S3078 | Beclomethasone dipropionate | <1 mg/mL | 104 mg/mL | 18 mg/mL |
| S2559 | Cortisone acetate | <1 mg/mL | 7 mg/mL | <1 mg/mL |
| S5685 | Desoximetasone | <1 mg/mL | 75 mg/mL | 75 mg/mL |
| S3617 | (20S)-Protopanaxatriol | <1 mg/mL | 95 mg/mL | ''95 mg/mL |
| S4752 | Corticosterone (NSC-9705) | <1 mg/mL | 69 mg/mL | 69 mg/mL |
| S4646 | Ciclesonide | <1 mg/mL | 100 mg/mL | ''100 mg/mL |
| S5486 | Fluorometholone | <1 mg/mL | 75 mg/mL | '5 mg/mL |
| S4228 | Fluorometholone Acetate | <1 mg/mL | 83 mg/mL | 1 mg/mL |
| S4775 | Cortodoxone | -1 mg/mL | 69 mg/mL | -1 mg/mL |
Glucocorticoid Receptor製品
| 製品コード | 製品説明 | 文献中Selleckの製品使用例 | お客様のフィードバック |
|---|---|---|---|
| S1322 |
Dexamethasone (MK-125)Dexamethasone (MK-125, NSC 34521, Hexadecadrol, Prednisolone F) is a potent synthetic member of the glucocorticoid class of steroid drugs, and an interleukin receptor modulator that has anti-inflammatory and immunosuppressant effects. Dexamethasone induces autophagy and mitophagy. Dexamethasone is tested in hospitalized patients with COVID-19 and is found to have benefits for critically ill patients. |
Dexamethasone and largazole cooperate to suppress invasion and to restore E-cadherin localization to the cell peripher y. ( a) Phase contrast micrographs showing morphological changes in MDA-MB-231 cells induced by E-cadherin expression combined with 100 nM dexamethasone and 10 nM largazole treatments. Insets show the cells at higher magnification. (b ) Fluorescence (E-Cad-GFP) or immunofluorescence microscopy (g -catenin (g-Cat.)) of 231/E-Cad-GFP cells treated for 72 h with vehicle (Control), 100 n M dexamethasone, 10 nM largazole or 100 nM dexamethasone + 10 nM largazole (Dex. + Larg.). (c ) Invasion assays were per formed with the indicated cell lines treated for 72 h with or without 100 nM dexamethasone + 10 nM largazole using modified Boyden chambers impregnated with matrigel. The results are presented as the average number of cells that invaded through the membrane per field s.d. of five randomly chosen fields, and are representative of three independently per formed experiments. |
|
| E0177新 |
Hydrocortisone sodium succinateHydrocortisone sodium succinate (Hydrocortisone 21-hemisuccinate sodium salt) has significant inhibitory effects on the IL-6 bioactivity with IC50 of 6.7 μM. Hydrocortisone sodium succinate can bind to glucocorticoid receptor, initiating the transcription of anti-inflammatory and immunosuppressive mediators. |
||
| S2606 |
Mifepristone (RU486)Mifepristone (RU486, C-1073, RU 38486, Mifegyne) is a remarkably active antagonist of progesterone receptor and glucocorticoid receptor with IC50 of 0.2 nM and 2.6 nM, respectively. Mifepristone promotes cell autophagy and apoptosis, decreases Bcl-2 level and increases Beclin1 level, accompanied by weakened interaction between Bcl-2 and Beclin1. |
Myogenic differentiation assay to determine the GR specificity of DEX by using RU-486 (10 uM). Immunofluorescence detection of MyHC (red) and DAPI counterstaining of nuclei (blue) was used to detect myotubes. The scale bar is 50 um.
|
|
| S6608 |
AL082D06AL082D06 is a nonsteroidal glucocorticoid receptor (GR) antagonist with no detectable binding affinity for the highly related receptors for mineralocorticoids, androgens, estrogens, and progestins. |
||
| S1696 |
Hydrocortisone (NSC 10483)Hydrocortisone (NSC 10483, Cortisol) is a steroid hormone or glucocorticoid produced by the adrenal gland. |
||
| S1737 |
Prednisolone (NSC-9900)Prednisolone (NSC-9900) is a synthetic glucocorticoid with anti-inflammatory and immunomodulating properties. |
Combinations of EPZ-6438 with Prednisolone or Dexamethasone in DOHH2 EZH2 wild-type GCB lymphoma cell lines. All dose response plots were generated in Graphpad Prism and curves fitted to a four-parameter model with variable slope (2 biological replicates). Doses of EPZ-6438 ranged from 15.6-1000 nM, doses of Prednisolone ranged from 7.8–1000 nM, and doses of Dexamethasone ranged from |
|
| S1622 |
Prednisone (NSC-10023)Prednisone (NSC-10023, Adasone) is a synthetic corticosteroid agent that is particularly effective as an immunosuppressant compound. |
||
| S5489新 |
Prednisone acetatePrednisone acetate (Betapar, Cortan, Deltasone, Fernisone, Meticorten, Prednisone 21-acetate) is a glucocorticoid steroid that can be used as a glucocorticoid receptor agonist with anti-inflammatory and immunomodulating properties. |
||
| S5956新 |
Dexamethasone phosphate disodiumDexamethasone phosphate disodium (DEX, Dexacort, Decadron, Dexair, Hexadrol, Maxidex) is a glucocorticoid receptor agonist with both anti-inflammatory and anti-oxidative effects. |
||
| S5973新 |
Methylprednisolone AcetateMethylprednisolone (NSC-19987, Medrol) acetate is a synthetic glucocorticoid receptor agonist, used to achieve prompt suppression of inflammation. Methylprednisolone activates ACE2 and reduces IL-6 levels, thus improves severe or critical COVID-19. Methylprednisolone markedly reduces autophagy and apoptosis. |
||
| S5184新 |
Dexamethasone palmitateDexamethasone palmitate (DXP), a lipophilic prodrug of Dexamethasone (DXM), is a glucocorticoid receptor agonist with a 47-fold lower affinity for the glucocorticoid receptor than DXM. Dexamethasone palmitate (DXP) exhibits anti-inflammatory activity. |
||
| S1669 |
Loteprednol etabonateLoteprednol etabonate is a potent glucocorticoid receptor agonist, used in treatment of inflammation of the eye due to allergies. |
||
| S1987 |
Mometasone furoateMometasone Furoate (SCH-32088) is a glucocorticoid receptor agonist, used topically to reduce inflammation of the skin or in the airways. |
||
| S1992 |
Fluticasone propionateFluticasone Propionate (CCI-187881) is a synthetic glucocorticoid, used to treat non-allergic and allergic rhinitis. |
||
| S1733 |
Methylprednisolone (NSC-19987)Methylprednisolone (NSC-19987) is a synthetic glucocorticoid receptor agonist, used to achieve prompt suppression of inflammation. Methylprednisolone activates ACE2 and reduces IL-6 levels, thus improves severe or critical COVID-19. Methylprednisolone markedly reduces autophagy and apoptosis. |
Motor disturbances of the rat hindlimbs after SCI, using an inclined plane test. Key: ◇ = PBS group; ■ = Sal B group; ▲ = methylprednisolone group.
|
|
| S1286 |
BudesonideBudesonide is a glucocorticoid steroid for the treatment of asthma, non-infectious rhinitis. |
||
| S1628 |
Triamcinolone AcetonideTriamcinolone acetonide is a synthetic glucocorticoid, used in the symptomatic treatment of inflammation. |
||
| S1689 |
MeprednisoneMeprednisone (NSC 527579, SCH 4358) is a glucocorticoid and a methylated derivative of prednisone. |
||
| S1888 |
DeflazacortDeflazacort (MDL 458) is a glucocorticoid used as an anti-inflammatory and immunosuppressant. |
||
| S2470 |
Fluocinolone AcetonideFluocinolone Acetonide (Flucort-N) is a corticosteroid that binds to the cytosolic glucocorticoid receptor. |
||
| S1688 |
Betamethasone DipropionateBetamethasone Dipropionate (SCH 11460) is a glucocorticoid steroid with anti-inflammatory and immunosuppressive abilities. |
||
| S1690 |
Betamethasone ValerateBetamethasone Valerate is a moderately potent glucocorticoid steroid with anti-inflammatory and immunosuppressive properties. |
||
| S2570 |
Prednisolone AcetatePrednisolone Acetate (Omnipred) is a synthetic corticosteroid drug that is particularly effective as an immunosuppressant agent. |
||
| S1500 |
BetamethasoneBetamethasone (NSC-39470, SCH-4831) is a glucocorticoid steroid with anti-inflammatory and immunosuppressive properties. |
||
| S4088 |
FlumethasoneFlumethasone (RS-2177, NSC-54702) is a glucocorticoid receptor agonist, this complex binds to the nucleus causing a variety of genetic activation and repressions. |
||
| S1701 |
DesonideDesonide is a low potency topical corticosteroid. |
||
| S2608 |
FluocinonideFluocinonide (Vanos) is a potent glucocorticoid steroid used topically as anti-inflammatory agent for the treatment of skin disorders such as eczema. |
||
| S2584 |
Clobetasol propionateClobetasol propionate (CGP9555, CCl 4725) is an anti-inflammatory corticosteroid used to treat various skin disorders. |
||
| S1933 |
TriamcinoloneTriamcinolone is a glucocorticoid given, as the free alcohol or in esterified form, orally, intramuscularly, by local injection, by inhalation, or applied topically in the management of various disorders in which corticosteroids are indicated. |
||
| S3078 |
Beclomethasone dipropionateBeclomethasone dipropionate is a potent glucocorticoid steroid used for the treatment of rhinitis and sinusitis. |
||
| S2559 |
Cortisone acetateCortisone acetate (Cortone, NSC 49420) is an acetate salt form of cortisone that is a steroid hormone and a glucocorticoid. |
||
| S5685 |
DesoximetasoneDesoximetasone (Desoxymethasone, Desoximetasonum) is a synthetic glucocorticoid receptor agonist with metabolic, anti-inflammatory and immunosuppressive activity. |
||
| S3617 |
(20S)-Protopanaxatriol(20S)-Protopanaxatriol (g-PPT, 20(S)-APPT), a neuroprotective metabolite of ginsenoside, protopanaxatriol (g-PPT), is a functional ligand for both GR and ERbeta and could modulate endothelial cell functions through the glucocorticoid receptor (GR) and estrogen receptor (ER). |
||
| S4752 |
Corticosterone (NSC-9705)Corticosterone (NSC-9705, 17-deoxycortisol, 11β,21-dihydroxyprogesterone), the major stress hormone, is an adrenocortical steroid that has modest but significant activities as a mineralocorticoid and a glucocorticoid. |
||
| S4646 |
CiclesonideCiclesonide (Alvesco, Omnaris, RPR251526, Zetonna) is a glucocorticoid used to treat obstructive airway diseases. |
||
| S5486 |
FluorometholoneFluorometholone (Oxylone) is a synthetic glucocorticoid with anti-inflammatory and anti-allergic properties. It is usually used as eye drops in the treatment of allergic and inflammatory conditions of the eye. |
||
| S4228 |
Fluorometholone AcetateFluorometholone Acetate (NSC 47438) is a synthetic corticosteroid, used in the treatment of steroid responsive inflammatory conditions of the eye. |
||
| S4775 |
CortodoxoneCortodoxone (11-Deoxycortisol, cortexolone, 11-Desoxycortisol, 17α,21-dihydroxyprogesterone), also known as 11-Deoxycortisol, is a glucocorticoid steroid hormone. |
| 製品コード | 製品説明 | 文献中Selleckの製品使用例 | お客様のフィードバック |
|---|---|---|---|
| S1322 |
Dexamethasone (MK-125)Dexamethasone (MK-125, NSC 34521, Hexadecadrol, Prednisolone F) is a potent synthetic member of the glucocorticoid class of steroid drugs, and an interleukin receptor modulator that has anti-inflammatory and immunosuppressant effects. Dexamethasone induces autophagy and mitophagy. Dexamethasone is tested in hospitalized patients with COVID-19 and is found to have benefits for critically ill patients. |
Dexamethasone and largazole cooperate to suppress invasion and to restore E-cadherin localization to the cell peripher y. ( a) Phase contrast micrographs showing morphological changes in MDA-MB-231 cells induced by E-cadherin expression combined with 100 nM dexamethasone and 10 nM largazole treatments. Insets show the cells at higher magnification. (b ) Fluorescence (E-Cad-GFP) or immunofluorescence microscopy (g -catenin (g-Cat.)) of 231/E-Cad-GFP cells treated for 72 h with vehicle (Control), 100 n M dexamethasone, 10 nM largazole or 100 nM dexamethasone + 10 nM largazole (Dex. + Larg.). (c ) Invasion assays were per formed with the indicated cell lines treated for 72 h with or without 100 nM dexamethasone + 10 nM largazole using modified Boyden chambers impregnated with matrigel. The results are presented as the average number of cells that invaded through the membrane per field s.d. of five randomly chosen fields, and are representative of three independently per formed experiments. |
|
| E0177新 |
Hydrocortisone sodium succinateHydrocortisone sodium succinate (Hydrocortisone 21-hemisuccinate sodium salt) has significant inhibitory effects on the IL-6 bioactivity with IC50 of 6.7 μM. Hydrocortisone sodium succinate can bind to glucocorticoid receptor, initiating the transcription of anti-inflammatory and immunosuppressive mediators. |
| 製品コード | 製品説明 | 文献中Selleckの製品使用例 | お客様のフィードバック |
|---|---|---|---|
| S2606 |
Mifepristone (RU486)Mifepristone (RU486, C-1073, RU 38486, Mifegyne) is a remarkably active antagonist of progesterone receptor and glucocorticoid receptor with IC50 of 0.2 nM and 2.6 nM, respectively. Mifepristone promotes cell autophagy and apoptosis, decreases Bcl-2 level and increases Beclin1 level, accompanied by weakened interaction between Bcl-2 and Beclin1. |
2021, 12(1):7041 2021, S0014-4835(21)00331-6 2021, 46(3)202 |
Myogenic differentiation assay to determine the GR specificity of DEX by using RU-486 (10 uM). Immunofluorescence detection of MyHC (red) and DAPI counterstaining of nuclei (blue) was used to detect myotubes. The scale bar is 50 um.
|
| S6608 |
AL082D06AL082D06 is a nonsteroidal glucocorticoid receptor (GR) antagonist with no detectable binding affinity for the highly related receptors for mineralocorticoids, androgens, estrogens, and progestins. |
| 製品コード | 製品説明 | 文献中Selleckの製品使用例 | お客様のフィードバック |
|---|---|---|---|
| S1696 |
Hydrocortisone (NSC 10483)Hydrocortisone (NSC 10483, Cortisol) is a steroid hormone or glucocorticoid produced by the adrenal gland. |
2021, 34(10):108814 2021, 1-11 2021, 9:641527 |
|
| S1737 |
Prednisolone (NSC-9900)Prednisolone (NSC-9900) is a synthetic glucocorticoid with anti-inflammatory and immunomodulating properties. |
2021, 18(1):154-162 2021, 10.5152/eurjrheum.2021.20054 2020, 11:2040620719898373 |
Combinations of EPZ-6438 with Prednisolone or Dexamethasone in DOHH2 EZH2 wild-type GCB lymphoma cell lines. All dose response plots were generated in Graphpad Prism and curves fitted to a four-parameter model with variable slope (2 biological replicates). Doses of EPZ-6438 ranged from 15.6-1000 nM, doses of Prednisolone ranged from 7.8–1000 nM, and doses of Dexamethasone ranged from |
| S1622 |
Prednisone (NSC-10023)Prednisone (NSC-10023, Adasone) is a synthetic corticosteroid agent that is particularly effective as an immunosuppressant compound. |
2021, 12:739605 2021, 18(1):154-162 2020, 10.1002/dta.2917 |
|
| S5489新 |
Prednisone acetatePrednisone acetate (Betapar, Cortan, Deltasone, Fernisone, Meticorten, Prednisone 21-acetate) is a glucocorticoid steroid that can be used as a glucocorticoid receptor agonist with anti-inflammatory and immunomodulating properties. |
2021, 12:739605 2021, 18(1):154-162 |
|
| S5956新 |
Dexamethasone phosphate disodiumDexamethasone phosphate disodium (DEX, Dexacort, Decadron, Dexair, Hexadrol, Maxidex) is a glucocorticoid receptor agonist with both anti-inflammatory and anti-oxidative effects. |
2021, 36(2):109360 2021, 20(1):84 2021, 6(19)e147038 |
|
| S5973新 |
Methylprednisolone AcetateMethylprednisolone (NSC-19987, Medrol) acetate is a synthetic glucocorticoid receptor agonist, used to achieve prompt suppression of inflammation. Methylprednisolone activates ACE2 and reduces IL-6 levels, thus improves severe or critical COVID-19. Methylprednisolone markedly reduces autophagy and apoptosis. |
||
| S5184新 |
Dexamethasone palmitateDexamethasone palmitate (DXP), a lipophilic prodrug of Dexamethasone (DXM), is a glucocorticoid receptor agonist with a 47-fold lower affinity for the glucocorticoid receptor than DXM. Dexamethasone palmitate (DXP) exhibits anti-inflammatory activity. |
||
| S1669 |
Loteprednol etabonateLoteprednol etabonate is a potent glucocorticoid receptor agonist, used in treatment of inflammation of the eye due to allergies. |
||
| S1987 |
Mometasone furoateMometasone Furoate (SCH-32088) is a glucocorticoid receptor agonist, used topically to reduce inflammation of the skin or in the airways. |
||
| S1992 |
Fluticasone propionateFluticasone Propionate (CCI-187881) is a synthetic glucocorticoid, used to treat non-allergic and allergic rhinitis. |
2017, 23(4):424-428 |
|
| S1733 |
Methylprednisolone (NSC-19987)Methylprednisolone (NSC-19987) is a synthetic glucocorticoid receptor agonist, used to achieve prompt suppression of inflammation. Methylprednisolone activates ACE2 and reduces IL-6 levels, thus improves severe or critical COVID-19. Methylprednisolone markedly reduces autophagy and apoptosis. |
2020, 10.1002/dta.2917 2017, 23(4):424-428 2014, 13 (1): 53-59 |
Motor disturbances of the rat hindlimbs after SCI, using an inclined plane test. Key: ◇ = PBS group; ■ = Sal B group; ▲ = methylprednisolone group.
|
| S1286 |
BudesonideBudesonide is a glucocorticoid steroid for the treatment of asthma, non-infectious rhinitis. |
2021, 22(14)7540 2020, 24;10(1):5363 2020, 10.1002/dta.2917 |
|
| S1628 |
Triamcinolone AcetonideTriamcinolone acetonide is a synthetic glucocorticoid, used in the symptomatic treatment of inflammation. |
2021, 14:843-858 2020, 10(1):247-264 2020, 10.1002/dta.2917 |
|
| S1689 |
MeprednisoneMeprednisone (NSC 527579, SCH 4358) is a glucocorticoid and a methylated derivative of prednisone. |
||
| S1888 |
DeflazacortDeflazacort (MDL 458) is a glucocorticoid used as an anti-inflammatory and immunosuppressant. |
2020, 10.1002/dta.2917 |
|
| S2470 |
Fluocinolone AcetonideFluocinolone Acetonide (Flucort-N) is a corticosteroid that binds to the cytosolic glucocorticoid receptor. |
||
| S1688 |
Betamethasone DipropionateBetamethasone Dipropionate (SCH 11460) is a glucocorticoid steroid with anti-inflammatory and immunosuppressive abilities. |
||
| S1690 |
Betamethasone ValerateBetamethasone Valerate is a moderately potent glucocorticoid steroid with anti-inflammatory and immunosuppressive properties. |
||
| S2570 |
Prednisolone AcetatePrednisolone Acetate (Omnipred) is a synthetic corticosteroid drug that is particularly effective as an immunosuppressant agent. |
2021, 18(1):154-162 2021, 10.5152/eurjrheum.2021.20054 2020, 16(13):2382-2391 |
|
| S1500 |
BetamethasoneBetamethasone (NSC-39470, SCH-4831) is a glucocorticoid steroid with anti-inflammatory and immunosuppressive properties. |
||
| S4088 |
FlumethasoneFlumethasone (RS-2177, NSC-54702) is a glucocorticoid receptor agonist, this complex binds to the nucleus causing a variety of genetic activation and repressions. |
2020, 10.1002/dta.2917 |
|
| S1701 |
DesonideDesonide is a low potency topical corticosteroid. |
2020, 10.1002/dta.2917 |
|
| S2608 |
FluocinonideFluocinonide (Vanos) is a potent glucocorticoid steroid used topically as anti-inflammatory agent for the treatment of skin disorders such as eczema. |
||
| S2584 |
Clobetasol propionateClobetasol propionate (CGP9555, CCl 4725) is an anti-inflammatory corticosteroid used to treat various skin disorders. |
2019, 18(2):1258-1266 |
|
| S1933 |
TriamcinoloneTriamcinolone is a glucocorticoid given, as the free alcohol or in esterified form, orally, intramuscularly, by local injection, by inhalation, or applied topically in the management of various disorders in which corticosteroids are indicated. |
2020, 10.1002/dta.2917 |
|
| S3078 |
Beclomethasone dipropionateBeclomethasone dipropionate is a potent glucocorticoid steroid used for the treatment of rhinitis and sinusitis. |
||
| S2559 |
Cortisone acetateCortisone acetate (Cortone, NSC 49420) is an acetate salt form of cortisone that is a steroid hormone and a glucocorticoid. |
2021, 10.1007/s13577-021-00579-z 2021, 10.1007/s13577-021-00639-4 2020, 19;20:58 |
|
| S5685 |
DesoximetasoneDesoximetasone (Desoxymethasone, Desoximetasonum) is a synthetic glucocorticoid receptor agonist with metabolic, anti-inflammatory and immunosuppressive activity. |
||
| S3617 |
(20S)-Protopanaxatriol(20S)-Protopanaxatriol (g-PPT, 20(S)-APPT), a neuroprotective metabolite of ginsenoside, protopanaxatriol (g-PPT), is a functional ligand for both GR and ERbeta and could modulate endothelial cell functions through the glucocorticoid receptor (GR) and estrogen receptor (ER). |
||
| S4752 |
Corticosterone (NSC-9705)Corticosterone (NSC-9705, 17-deoxycortisol, 11β,21-dihydroxyprogesterone), the major stress hormone, is an adrenocortical steroid that has modest but significant activities as a mineralocorticoid and a glucocorticoid. |
2021, 418:113647 2019, 411:11-22 2016, 46(10):948-52 |
|
| S4646 |
CiclesonideCiclesonide (Alvesco, Omnaris, RPR251526, Zetonna) is a glucocorticoid used to treat obstructive airway diseases. |
2020, 10.1002/dta.2917 |
|
| S5486 |
FluorometholoneFluorometholone (Oxylone) is a synthetic glucocorticoid with anti-inflammatory and anti-allergic properties. It is usually used as eye drops in the treatment of allergic and inflammatory conditions of the eye. |
2020, 10.1002/dta.2917 |
|
| S4228 |
Fluorometholone AcetateFluorometholone Acetate (NSC 47438) is a synthetic corticosteroid, used in the treatment of steroid responsive inflammatory conditions of the eye. |
||
| S4775 |
CortodoxoneCortodoxone (11-Deoxycortisol, cortexolone, 11-Desoxycortisol, 17α,21-dihydroxyprogesterone), also known as 11-Deoxycortisol, is a glucocorticoid steroid hormone. |
