• C-Raf/Raf-1
  • B-Raf
  • A-raf

A-raf 阻害剤

製品コード 製品名 製品説明 Selective / Pan IC50 / Ki
S7926 Lifirafenib (BGB-283) Lifirafenib (BGB-283, Beigene-283) potently inhibits RAF family kinases and EGFR activities in biochemical assays with IC50 values of 23, 29 and 495 nM for the recombinant BRAFV600E kinase domain, EGFR and EGFR T790M/L858R mutant. Pan WT A-RAF, IC50: 1 nM