H3 receptor Selective 阻害剤 | 拮抗剤

製品コード 製品名 製品説明 Selective / Pan IC50 / Ki
S2813 Ciproxifan Ciproxifan is a highly potent and selective histamin H3-receptor antagonist with IC50 of 9.2 nM, with low apparent affinity at other receptor subtypes. Selective Histamine H3 receptor, IC50: 9.2 nM
S3176 Betahistine 2HCl Betahistine is a histamine H3 receptors inhibitor with IC50 of 1.9 μM. Selective Histamine H3 receptor, IC50: 1.9 μM
Tags: H3 receptor inhibitor | H3 receptor cancer | H3 receptor activation | H3 receptor activity | H3 receptor phosphorylation | H3 receptor mutation