H3 receptor Selective 阻害剤 | 拮抗剤
||Selective / Pan
||IC50 / Ki
||Ciproxifan is a highly potent and selective histamin H3-receptor antagonist with IC50 of 9.2 nM, with low apparent affinity at other receptor subtypes.
||Histamine H3 receptor, IC50: 9.2 nM
||Betahistine is a histamine H3 receptors inhibitor with IC50 of 1.9 μM.
||Histamine H3 receptor, IC50: 1.9 μM
Tags: H3 receptor inhibitor | H3 receptor cancer | H3 receptor activation | H3 receptor activity | H3 receptor phosphorylation | H3 receptor mutation