PPARγ 選択性阻害剤 | 作動薬 | 拮抗剤
|製品コード||製品名||製品説明||Selective / Pan||IC50 / Ki|
T0070907 is a potent and selective PPARγ inhibitor with IC50 of 1 nM, with a >800-fold selectivity over PPARα and PPARδ.
|Selective||PPARγ, IC50: 1 nM|
Rosiglitazone, a member of the thiazolidinedione class of antihyperglycaemic agents, is a high-affinity selective agonist of the peroxisome proliferator-activated receptor-γ.
|Selective||PPARγ, IC50: 42 nM|
Pioglitazone is a selective peroxisome proliferator-activated receptor-gamma (PPARgamma) agonist, used to treat diabetes.
GW9662 is a selective PPAR antagonist for PPARγ with IC50 of 3.3 nM, with at least 100 to 1000-fold functional selectivity in cells with PPARγ versus PPARα and PPARδ.
|Pan||PPARγ, IC50: 3.3 nM|
FH535 is a Wnt/β-catenin signaling inhibitor and also a dual PPARγ and PPARδ antagonist.
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