Selective 阻害剤 | 作動薬 | 拮抗剤

製品コード 製品名 製品説明 Selective / Pan IC50 / Ki
S2103 Naltrexone HCl Naltrexone HCl is an opioid receptor antagonist with IC50 of 8 nM used primarily in the management of alcohol dependence and opioid dependence. Selective opioid receptor, IC50: 8 nM
S3204 Meptazinol HCl Meptazinol is a unique centrally active opioid analgesic, which inhibits [3H]dihydromorphine binding with IC50 of 58 nM. Selective
S2503 Racecadotril Racecadotril is a peripherally acting enkephalinase inhibitor with an IC50 of 4.5 μM Selective
S3066 Naloxone HCl Naloxone HCl is an opioid inverse agonist drug used to counter the effects of opiate overdose. Selective
S2480 Loperamide HCl Loperamide HCl is an opioid-receptor agonist with an ED50 of 0.15 mg/kg. Selective
S1139 ADL5859 HCl ADL5859 HCl is a δ-opioid receptor agonist with Ki of 0.8 nM, selectivity against opioid receptor κ, μ, and weak inhibitory activity at the hERG channel. Phase 2. Pan μ-opioid receptor, Ki: 32 nM